ZempiloAmalungiselelo

Imiyalelo yokusebenzisa "klopiksol" inkcazo ichiza, izigxeko

Yintoni na le neziyobisi "klopiksol '? ncomo Consumer neempawu eli chiza ziya kuqwalaselwa izinto kweli nqaku.

Ifom ye yokulungiselela, ukwakheka, inkcazelo, ukupakishwa

Kwezi mali kufuneka iifom ukukhululwa ezahlukeneyo. Sinikela ngoku.

1. "klopiksol" - iipilisi lipholi pink, umbala epinki-brown kwaye zifuna ukuba ngqombela-brown (2 mg, 10 mg-25 mg, ngokulandelelanayo). Ba setyhula kwaye lenticular imilo, kunye film ngeso lenyama.

Into esebenzayo ye sisixhobo zuclopenthixol dihydrochloride. Kwakhona, kuba iqulathe 85% glycerol, iitapile starch, copovidone, monohydrate lactose, microcrystalline kwincindi, talc, nemagnesium stearate, neoli, hydrogenated kukaCastor.

Ekuthengisweni ithathwa beziyobisi iza kwimigqomo zeplastiki kunye neebhokisi ezenziwe ikhadibhodi.

2. Isisombululo ioli / m "klopiksol". Ukuphonononga bathi esi sixhobo kuthengiswa ampoules ezenziwe ngeglasi enemibala. Isisombululo ngokwayo inombala bulubhelu elubala. Akanalo kwaphela ngamasuntswana.

Into esebenzayo yale imithi decanoate zuclopenthixol. Kwakhona le nkqubo ibandakanya triglycerides.

Amayeza isenzo "klopiksol"

medicament kubhekwe yemvelaphi thioxanthene - a neuroleptic. Yena imiphumo ethile inhibitory kunye antipsychotic. Ukongeza, le isixhobo ibonisa okulalisa.

A ulawulo elinye ichiza kunegalelo Akuhlangani ngokukhawuleza iimpawu ngengqondo. iimpawu sine ye ichiza babonakaliswa emva kweeyure ezi-2, kunye nefuthe layo ngokubanzi buhlala iintsuku ezi-3.

iimpawu entshukumo yokulungiselela

Ngokutsho kweengcali, inaliti yale Isisombululo kuyacetyiswa ukuphumeza lamathuba (kwiiveki-4).

Emva ulawulo ngomlomo, incopho xiyimiso iziyobisi afunyenwe emva 4 h. Zuclopenthixol bioavailability imalunga 44%.

Emva ulawulo intramuscular kwento esisiseko yale amalungiselelo phantsi cleavage enzymatic. Oku kuvelisa acetic acid kunye zuclopenthixol esebenzayo. Icandelo lokugqibela izixa ezincinane kwazona ngobisi lwebele kwaye ingena isithintelo placental.

Xa ukufumana amayeza zibe kwixesha isiqingatha ubomi layo eziyi-20. It ubonisa kakhulu endleni kwaye ngokuyinxenye - kunye nomchamo.

Ubungqina obubonakalayo buxela ukuba ukusetyenziswa

Kwezinye iimeko, ichiza emiselweyo kwizigulana ingqalelo? Oko ikuthethayo ngalo imiyalelo ukusetyenziswa? "Klopiksol" kuboniswe:

  • schizophrenia acute kunye ezingapheliyo kunye nezinye izifo zengqondo, kuquka ezo iimfeketho zokufeketha ebandakanya (paranoid), nemibono kunye nokuphazamiseka kwindlela yokucinga;
  • imo kukuphazamiseka, ubutshaba, ixhala (eziphakamileyo), ubuvila;
  • ukukhubazeka engqondweni, nto leyo kudityaniswe kukuphazamiseka, kukuphazamiseka (lengqondo), kunye nezinye izifo e zokuziphatha;
  • mania of njengemanic-depressive;
  • dementia saka, nokudideka, ukuziphatha kakuhle, iingcamango usoyika kwaye nochuku.

Siphelisa imithi ukusetyenziswa

ukuba asebenzise nini na neuroleptic ingxelo? Oko ikuthethayo ngalo imiyalelo ukusetyenziswa? "Klopiksol" into contraindicated ku:

  • ukunxila acute kunye barbiturates;
  • etsolo uhlobo ukunxila okanye utywala;
  • analgesics ukunxila etsolo (opioid).

Kufuneka kuqatshelwe ukuba uthe arhente antipsychotic alisetyenziswa sikarhulumente comatose.

Imiyalelo yokusebenzisa

"Klopiksol" Amacwecwe athathwa ngomlomo. Le umthamo eli chiza ikhethiwe ngamnye ngokuxhomekeke imeko yesigulane. Ekuqaleni unyango ngamachiza ilawulwa ngeedosi ephantsi, uze ngokukhawuleza banda isiphumo yabo clinical.

Xa yabonisa eliphakathi kunye nezigulo zengqondo lokuqala idosi "klopiksol" yi-20 mg ngosuku. Ukuba kuyimfuneko, oko kwandiswa ukuya mg-20.

Xa schizophrenia etsolo episode kunye nezinye izifo zengqondo, indalo etsolo, mania kwaye yababuhlungu iyeza ukuphazamiseka idosi ichanekile 10-50 mg ngosuku.

Xa ezingapheliyo States ngengqondo uhlobo, kwakunye ngesifo kunye nezinye kwengqondo, idosi ingqalelo nokuxhasa esebenzisa 20-40 mg ngosuku.

Xa ukuphazamiseka kubantu abane ukukhubazeka idosi yengqondo 6-20 mg ngosuku. Ukuba kuyimfuneko, oko kwandiswa ukuya 25-40 mg ngosuku.

Xa izifo saka kukuphazamiseka nochuku eli chiza ibhalwa ne nedosi ye-2-6 mg ngosuku. Ukuba kuyimfuneko, isixa ezichaziweyo ichiza lanyuka ukuya 10-20 mg ngosuku.

Umthamo isisombululo oyile

Ndifanele kungena njani isisombululo yeoli? Yintoni le usixelela yesikhokelo? "Klopiksol 'elawulwa ngohlobo anzongonzongo / ziphene m oluqhutywa kummandla gluteal.

Imali obacetyiswayo ngenaliti enjalo kufuneka 1-3 ml. Ukuba kuyimfuneko, ngokuphindaphindiweyo iinaliti ezenziwe emva kwesithuba seentsuku ezi-3. Ezinye kwizitofu izigulane abongezelelweyo baqeshwa emva kosuku okanye ezimbini.

sequela angafuneki

Yiyiphi indlela ezimbi ebangela ichiza "klopiksol"? iziphumo ebezingalindelekanga eli chiza kuqhelekile kakhulu. Ezi ziquka oku kulandelayo:

  • ukugcinwa wokuchama, ccomodation;
  • Iimpawu extrapyramidal (kwisigaba sokuqala unyango), ukozela;
  • tachycardia, isiyezi, hypotension intolerance ;
  • zeDyskinesia tardive (unyango elide);
  • kwesisu, umlomo owomileyo, utshintsho ezidlulayo kwiimvavanyo umsebenzi esibindini.

amacala libanda

isiqaqa, ukozela, unditsho,: Ngenxa libanda, le mali, ezi mpawu zilandelayo sifo extrapyramidal, athuke, hypotension, esihanahanisa- okanye nokushisa.

Ukuze ukususa isimo isigulane wahlanjwa esiswini nokunika sorbents. Kwakhona, kwanonyango inkxaso nomqondiso.

imithi

Ukulungiselela "klopiksol" (10 mg) iphucula okulalisa utywala, barbiturates kunye nezinye iziyobisi leyo ibe nesiphumo inhibitory kwi-CNS.

Eli chiza kufuneka zidityaniswe kunye guanethidine neziyobisi kunye neziphumo ezifanayo ngenxa kunokwenzeka yokuvimba ifuthe labo umfutho.

ukwamkelwa ngaxeshanye nabo "klopiksol" kungacutha ukusebenza arhente adrenergic, kuquka "Levodopa".

Xa kudityaniswe iindlela njenge "piperazinyl" yaye "MCP" kwandisa umngcipheko iimpawu extrapyramidal.

izincomo ezithile

Drug "klopiksol", ixabiso oboniswe apha ngezantsi, kunye isilumkiso emiselweyo kubantu abanesifo sentliziyo, kohlobo, kunye nezigulo convulsive.

unyango elide kufuneka ibe esweni rhoqo clinical ukuhlola imeko yesigulane.

Xa efumene neuroleptics CSN banokuba yingozi. Ezona mpawu ziphambili karhulumente ezinjalo ngqongqo dystrophy, ukuphazamiseka osezingqondweni, kwekhono of NS yawo, komzimba.

Iindleko ukulungiselela kwakhona ngayo

Price ingqalelo ichiza ixhomekeke kwifom release. 2 amacwecwe mg kwi isixa lamaqhosha-50 zimalunga 250 engange, 25 mg (iiyunithi 100) - malunga ne-1600 engange, no-10 Amacwecwe mg (iziqwenga 50) - malunga ne-480 engange.

Ngokumalunga isisombululo oyile, ixabiso layo lifike 2300 engange.

Amaninzi, ezo ncomo yabathengi yokulungiselela 'klopiksol "ushiye ezo izigulane kusetyenziswa ichiza ngokohlobo ngenaliti. izigulane ezinjalo bathi izinga isicelo esi sixhobo Kulula kakhulu ukuyisebenzisa. Oku kungenxa yokuba izitofu kufuneka kwenziwe enqabile (njengoko kuchasiwe uthatha iipilisi).

Ngokutsho ingxelo yabathengi, ichiza "klopiksol" i antipsychotic kakuhle kakhulu kwaye fast-ngokwenza. Kodwa ke, ngelishwa, oko kudla ibanga iziphumo ebezingalindelekanga.

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