ZempiloAmalungiselelo

Ichiza "Betaxolol": imiyalelo ukusetyenziswa, inkcazo, ukwakhiwa kunye nohlolo

Amathontsi kuba amehlo "Betaxolol" (yemiyalezo yahlula kubo njengoko uyakhetha beta-blocker elide action) zisetyenziswa lwamehlo ndlela, nezidanga ezisetyenziswa ekunyangeni ezahlukeneyo sentliziyo izifo.

ifomu Release komsindo

Lithetha "Betaxolol" evela ngokohlobo amacwecwe kunye wamehlo. Enye tablet emhlophe nala ukutyabeka umboniso equlathe 20 mg Isithako esisebenzayo betaxolol hydrochloride. Njengoko izinto ezongezelelweyo zezi: carboxymethylstarch sodium, nemagnesium stearate, microcrystalline kwincindi, monohydrate lactose, aerosil. UKwakhiwa yeqokobhe iquka Polyvinyl utywala, Opadry emhlophe 2, macrogol, talc, titanium dioxide.

Wapakisha iziqwenga ezili-10 ngo-aluminiyam namadyungudyungu iipilisi "Betaxolol." Imiyalelo ukusetyenziswa livalelwe kwibhokisi yekhadibhodi.

Kwi-drop iliso nganye 1 ml akhawunti 5.6 mg Isithako esisebenzayo betaxolol hydrochloride. izinto Secondary eliquka mithi: hayidroksayidi sodium, benzethonium chloride, zehydrochloric acid, dihydrate, disodium edetate, isodiyam chloride, amanzi. Le into elityheli ngaphaya. Ewiliko iye ifakwe kwibhotile-IV (5 okanye 10 ml). lingatshajiswanga ngakumbi yaye dropper ityhubhu kwi umthamo 1.5-5 ml. Xa ibhokisi yekhadibhodi waza wabeka imiyalelo ibhotile-dropper.

Aphezulu ubomi ezikhabhathini

Impilo iziyobisi (tablets kunye wamehlo) yiminyaka emithathu. Emva kokuvula i-ibhotile ngamathontsi kunokugcinwa akukho ngaphezu kweentsuku ezingamashumi amabini anesibhozo.

Pharmacokinetics

Isenzo amayeza beziyobisi luphawulwa beta-uyakhetha adrenoblokiruyuschey, antianginal, umfutho, antiarrhythmic, antiglaucoma yokuqhelaniswa nezifundo.

ezenza Iibhloko beta1-adrenergic Umsebenzi sympathomimetic, kananjalo olungaphaya iipropati ezincinane ndizayo ozinzileyo. Kunciphisa susceptibility izicwili ukuba catecholamines, Azeke esembindini iminqweno, ime i secretion of renin. Oku kunciphisa izinga lentliziyo kunye kunciphisa ukusetyenziswa ioksijini engabalulekanga (iipropati antianginal). Iibhloko zenzeka nakujoliso olutsha ethunjini kwi imithambo, AV-ezihamba kunye.

Isiphumo emsebenzini emva kweeyure ezimbini emva kokungenisa, nengqwalaselo iziyobisi ubuninzi emzimbeni busisigxina ngeeyure 3-4 kwaye ithatha iiyure 12-24 usebenziso rhoqo eqhelekileyo ichiza iintsuku 7-14. It likhusela ngokuchaseneyo ukunyuka koxinzelelo lwegazi ngethuba umthambo noxinezeleko nasengqondweni.

Unyango lwe soxinzelelo lwegazi kungenxa ekuphungulweni ventricular mass yasekhohlo kunye nokwandisa umsebenzi wayo contractile. Malunga ne-75% ezigulane abangeva ukumodareyitha lwegazi ukuphendula kakuhle ukuya monotherapy onjalo. ukusetyenziswa elide ichiza aluchaphazeli ngokulinganayo of lipid ukutya kunye kukhuthaza sodium. Xa abantu abane sisifuba nokukrala ngendlela ezigulo ezondeleyo akuthethi ukunciphisa ukusebenza kwemiphunga.

Wamehlo "Betaxolol" (manual imfundiso ithi malunga impembelelo ichiza ukunciphisa uxinzelelo intraocular ngokunciphisa ulwelo intraocular) musa ukuba iziphumo ebezingalindelekanga ezifana namhla-ubumfama, miosis, spasm zokuhlala, kunye nombono luzizi.

Le nguqu kuphunyelelwa emva isiqingatha seyure emva kokuba isicelo, i ndzo ubuninzi baqaphela emva kweeyure ezimbini kwaye ithatha iiyure ezilishumi elinesibini.

Ubungqina obubonakalayo buxela ukuba ukusetyenziswa

Acetyiswayo lokufunyaniswa "lwegazi" fit ehlala abantu ischaemia engabalulekanga (angina), akathisia, nomsindo neuroleptics, "Betaxolol" iipilisi.

Eyedrops (yemiyalezo ukuba ubonane nogqirha ngaphambi kokuba uyisebenzise) kubonisiwe kwi isifo engile evulekileyo neglaucoma, hypertension intraocular. Amagqirha amisele ichiza emva laser trabeculoplasty. Used in kunyango umfutho ixesha elide, imfuneko ezivele ngenxa ungenelelo lwamehlo yotyando.

Izimo medical

Nangona ukusebenza engqiniweyo "Betaxolol" iziyobisi (Usetyenziso Drug bacetyiswa ukuba bagcine ngokungqongqo pamo emiselwe ngugqirha hayi self-medicate), ukusetyenziswa kwalo Izimo ezithile. Ezi ziquka hypersensitivity yecandelo esebenzayo beziyobisi, kwaye izinto ezongezelelweyo kumafa yayo. Kwakhona engavunyelwa xa fikisruyutsya sinus bradycardia (ngaphantsi kwe 45-50 u. / Min) kunye sinus abagulayo. Awukwazi ukusebenzisa iyeza kwi AV yaye kuvalwe II-III isidanga, hypotension. Contraindicated "Betaxolol" abantu ngokothuka cardiogenic kwizigulane kunye ukusilela ngentliziyo kakhulu kwaye yababuhlungu ukusilela obstructive zemiphunga.

Kufanele kuthathwe kwizigulane kunye nenyumoniya ezingapheliyo, izigulane angina ezingazinzanga, kukho ukuthambekela bradycardia. Ahlale evule amehlo kufuneka kwenze AV-block I degree, ukusilela neuropathy kwegazi. Kufuneka ube izigulane ingakumbi Qhaphela xa seswekile, hypoglycemia, isibindi kunye nesifo sezintso, hyperthyroidism. Oogqirha kufuneka esweni amayeza xa izigulane nobuthathaka kwezihlunu abadala kunye nabantwana.

Ngethuba lokukhulelwa lokwaphusa iziyobisi ukuthatha, ukuba inzuzo ezilindelekileyo ukuya unina komonakalo ingozi olungekazalwa. Ngexesha unyango kufuneka ayeke ibele-lwebele.

"Betaxolol": imiyalelo yokusebenzisa

Price, ukubuyekeza, abasebenzi - ezi izinto ezintle iziyobisi ezibangela izigulane ukuba ngokuphindaphindiweyo ukuze uyikhethe.

Ezi tablets kufuneka enxila kusasa. dragees lwegazi bazithathe kanye, kuqalwa umthamo we-10 mg. Ukuba emva kweveki akufani ziphumo zinqwenelekayo ifunyenwe, ithamo landiswa ukuya ml-20. Ukuba isiphumo kulindeleke ayiphumelelanga kwakhona ukufikelela, ngoko emveni kweentsuku 7-14, ukwandisa ithamo ku-40 mg.

Izigulane umsebenzi kakuhle kidney, dialysis, kwakunye abadala kufuneka basebenzise amayeza isixa-5 mg kanye yonke imihla. Ukuba kuyimfuneko, ithamo angandiswa zonke iintsuku ezili-14 ngo-5 mg. Lucebisa ukuba ingagqithi idosi iphezulu - ml 20 "Betaxolol" ukulungiselela - imiyalelo ukusetyenziswa.

Abstract icebisa ukusebenzisa wamehlo glaucoma. Instillation kufuneka wenziwe ngokungqongqo lo sac conjunctival. A idosi enye ngomnye ukuhla. Esi siganeko kwenzeka kabini ngemini. Kwinyanga yokuqala yonyango, ugqirha kufuneka iliso uxinzelelo intraocular yesigulana.

imiphumela emibi

Amabango nesiphumo esibi iziganeko yesicelo "Betaxolol" ukulungiselela imfundo manual. Ixabiso ichiza yedemokhrasi, nto leyo eyenza kube lula ukuba onke amacandelo oluntu (80 miri. Kuba 5 ml igutyana kunye 370 engange. Kuba amacwecwe 30).

Ngexesha unyango "Betaxolol" kusenokubakho chronic fatigue kunye intloko ebuhlungu, isiyezi, ukozela, sokulibala, ixhala, ukudandatheka. Ukuncipha ingqondo, amabi, nemibono, kunesifo, neuralgia, ukuphazamiseka vestibular.

Ezinye izigulane ziye ibonwe kwaye ukuchama induku ukungathobeli, iintlungu emabeleni (e abafazi), prostatitis, utshintsho ibele fibrocystic. Kwakukho ukuqunjelwa, urhudo, umlomo owomileyo, isicaphucaphu, ukugabha, ukuqhina, iintlungu esiswini. Ichiza ngamanye amaxesha ngokungalunganga kuchaphazela nesifo semiphunga ezosulelayo, dyspnea, ibangela iintlungu esifubeni, pharyngitis, nokuthimliswa, sinusitis. bronchospasm Fixed, dyspnea, ukusilela sokuphefumla.

Phakathi imiphumela sele ezikhethelwe ngolu hlobo lulandelayo: bradycardia, hypotension, engabalulekanga iposi, nesifo sentliziyo, leukocytosis, thrombocytopenia purpura kunye nezinye izifo. Kwanele kunqabile arthralgia, tendonitis, myalgias.

Ingaba irhashalala, alopecia, negazi, nangokhwekhwe, utshintsho ubunzima bomzimba, erythema, emzimbeni, exacerbation of ukhwekhwe, hypertrichosis, prurigo.

Ukusetyenziswa wamehlo uyakwazi ukuba bawaphikise lacrimation, amehlo ezomileyo, ukungaboni, photophobia, keratitis, erythema, umzimba angaphandle imvakalelo emehlweni, uvakalelo kwenwebu yamehlo, anisocoria kunye photophobia.

oyi

Xa Betaxolol drug therapy (umyalelo kwi isicelo iinkcukacha idosi indlela zonyango) kudla utshintsho parameters elebhu. Kusenokuba yokusabela lobuxoki eyakhayo dope, ukwanda titers omzimba antinuclear kunye t. D.

Libanda, "Betaxolol" iziyobisi

Imiyalelo yokusebenzisa (analogs babe into efanayo esebenzayo yaye kunempembelelo efanayo) licebisa ngamandla idosi. Kungenjalo, nazo iimpawu ezingemnandi ezifana:

  • nesiyezi;
  • ephula yegazi;
  • bronchospasm;
  • hliswa glucose igazi;
  • amahlaba imisipha;
  • lungasebenzi.

Kule meko unyango classical ababelwe ngolu hlobo lulandelayo:

  • lavage esiswini;
  • sebenzisa kwezinto izifunxi;
  • unyango lingaze - atropine efakwa 1-2 mg ibeta-agonists, nadlamkisayo agents, igazi iziyobisi;
  • ngexesha emalithathwe ukufundisa transvenous (wabelwa kuphela kwiimeko ezingxamisekileyo).

izinyathelo Personal

Therapy kufuneka kwenziwe phantsi kweliso elibukhali likagqirha. Xa unyango akakwazi phawula lokuqala inqanaba hyperthyroidism kunye hypoglycemia. Oku eqhelekileyo kwizigulane kunye seswekile. Ukuncipha iinkqubo zembuyekezo iimpahla sentliziyo kunye negazi. Awukwazi ukusebenzisa ichiza phambi uqhaqho.

ukusetyenziswa rhoqo kweziyobisi abakhulileyo kwandisa umngcipheko emzimbeni, imeko yengqondo ukutshabalala, ukuphazamiseka umsebenzi sentliziyo. Izigulane isifo sezintso zesibindi kufuneka abe phantsi kweliso likagqirha iintsuku ezine zokuqala. Ukuba Imbali zokwalana kungenzeka ukwandisa hypersensitivity nokunciphisa isiphumo nezinyangayo adrenaline.

Xa ukusetyenziswa kweziyobisi kungavumelekanga ukuba iziselo ezinxilisayo. Kwakhona Awukwazi yokuvele ukuyeka unyango kwaye kufuneka ukwenze oko kancinane, ngokunciphisa idosi kwisithuba seeveki ezimbini. Ucebisa abaqhubi ukuba balumke xa ukusetyenziswa kwamayeza "Betaxolol" umyalelo manual.

Price, analogue beziyobisi

Ukuba ichiza anisondelanga, ugqirha angasoloko sinikele analog, nto leyo ngokufuthi kwahluka kuphela ixabiso. Ngenxa yoko, amacwecwe kunye ilahla "Betaxolol" iindleko malunga 80-370 engange. Ngu analogue amacwecwe ziquka:

  • "Betacam" (waseSipro), kubiza imali engange malunga 300 tablet-20.
  • "Lokren" (France), ixabiso tablet 28 - 600-700 engange, kwaye nangeepilisi 56 - 1000-1200 engange.

Wamehlo nge hydrochloride betaxolol into esebenzayo indawo yimithi zilandelayo:

  • "Betalmik EU" (Slovakia), 160-200 engange.
  • "Betoptik" (Belgium, eUnited States), malunga 300 engange.
  • "Betoptik C" (Belgium, USA), ngaphakathi engange-300.
  • "Betoftan" (saseRomania), 200 engange.
  • "Ksonef" (India), 180 engange.
  • "Ksonef BC" (India), malunga 150 engange.
  • "Optibetol" (Poland).

Uthi malunga ukusebenza yonyango lwegazi iziyobisi "Betaxolol" umyalelo manual. Price, reviews (analogue ayabiza, kodwa isiphumo esifanayo emzimbeni) - lonke olu lwazi lunikezelwa kweli nqaku.

Views ezigulane

Lucebisa ukusetyenziswa "Betaxolol" imenyu in lwamehlo manual therapy lokufundisa. Intengo (reviews athi le yenye ngeengenelo beziyobisi) iphantsi, yaye ukuze bakwazi ukuthenga phantse naluphi abadinga unyango. Izigulane ezininzi zibeka nokunyamezela ezilungileyo wamehlo. Bathi ukuba ndingamkhubekisi iziphumo ebezingalindelekanga. Isiphumo nokubonakala kwawo ekupheleni kweveki yokuqala.

Ngoncedo iipilisi zabantu ukulawula uxinzelelo lwegazi. Ichiza inceda ukwehlisa umthwalo entliziyweni, kuphucula imeko jikelele zezigulane. Abanye stress disorder inkqubo ukwetyisa ngemihla ekuqaleni ukuthatha iipilisi. Kukho abantu awanikeleyo ichiza iye yabangela irhashalala komzimba kwaye bomvu apha esikhumbeni. Umntu waphawula isicaphucaphu kunye arrhythmia kakhulu.

Uninzi ukubuyekeza iyeza ezintle, izigulane ziye iyahlutha le unyango.

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