Zempilo, Amalungiselelo
"Antabuse" iipilisi. Ukuphononongwa, guide ixabiso
Oku kubizwa etywaleni sisifo amagama nomkhwa Ethanol kunye ukuxhomekeka ngokwasemzimbeni nangokwasengqondweni kuyo. Olu hlobo kakubi. Kule meko, ukulahlekelwa lulawulo phezu isixa basela utywala kwandisa ukunyamezelana kuyo (ukufezekisa utywala ulwaneliseko rhoqo ithamo ukwandisa) kunye syndrome zokurhoxa kwenzeka, ichaphazela izibilini kuvela memory iyaphelelwa.
Izigulane unengxaki yokusela, ekuthiwa otywala. Mphathe sifo kufuneka engqondweni nasemzimbeni. Amaxesha amaninzi, oogqirha amisele eli chiza kubantu "Antabuse". Imiyalelo zokusetyenziswa, amaxabiso amayeza, reviews zonyango ziboniswa apha ngezantsi.
Nokupakisha, imilo, kunye nenkcazo isakhiwo
Koko benza ichiza buthengiswa "Antabuse"? Baqinisekiswa ingxelo ukuba iyeza enjalo zingathengwa ngohlobo, amacwecwe effervescent ngeenxa emhlophe. Ba tyaba, ngohlangothi beveled, umngcipheko kwakunye iphawulwe «CD» kunye «C» kumacala ahlukeneyo iingozi.
Ukubunjwa olu nyango ziquka disulfiram. Ngaphandle kwalo, ukulungiswa iqulethe ingqolowa starch, povidone, isodiyam hydrogencarbonate, tartaric acid, colloidal lesilicon dioxide, talc, microcrystalline neselulosi kunye wemagniziyam stearate.
Tablets "Antabuse" zibekwe kwizikhongozeli zeplastiki Imiqulu kwikhadibhodi.
iimpawu pharmacodynamic
Yintoni na ichiza "Antabuse"? Manual ukuba oku kuthetha antialcoholic. It abangaphangeliyo acetaldehyde dehydrogenase, nto leyo ebandakanyekileyo nethe-ethanol. Usenokubeka elinye ixesha inkqubo yayo igcwala ebangela ukuqokelela kotywala kunye nophuhliso kunxilwe olunamandla, kulandele iimvakalelo enzima njenge iintlungu throbbing kunye nesandi entloko, tachycardia, palpitation, ukwehliswa uxinzelelo lwegazi, isicaphucaphu, ukungaboni kunye nokugabha.
Ngokutsho kweengcali, ezi mpawu ezingemnandi igalelo kuphuhliso lokunyamezela moya reflex utywala.
iipropati pharmacokinetic
njani kukufakwa "Antabuse 'iziyobisi? Manual ibonisa ukuba ichiza wendele yi 70-80%. Yena enyibilikayo kakhulu lipids kwaye ithande ukuba yande kwindawo ngamanqatha.
Le into esebenzayo yomenzeli umzimba ngokukhawuleza kakhulu, kwaze oko kwakhokelela metabolite uguqulwa - Ester imethyl dietiltiokarbaminovoy acid. Its lamanani igazi eliyincopho kumiselwa emva 4 h. Nangona umsebenzi ngokunxulumene acetaldehyde dehydrogenase elifana neli kuphela emva kweentsuku ezintathu.
Isiqingatha-wobomi ichiza iiyure ezili-10. Ngaphezu koko, umsebenzi wayo xa kuthelekiswa aldehyde dehydrogenase isaqhubeka elide kakhulu. Ngoko ke, emva kokuba yokurhoxiswa isiphumo amacwecwe kuvandlakanywa okwelinye iintsuku 7-14.
Ichiza livela umchamo, yaye ngokuyinxenye ngenxa amathumbu kunye umoya.
ubungqina
Kwezinye iimeko, siyobisi ngempumelelo liziphatha "Antabuse"? Ukuphonononga baxele ukuba eli ziko isetyenziswa ngokubanzi nokuthintela ukuhluleka kwi ukunyanga ukuxhomekeka utywala kunye butywala.
Izimo
Xa kufuneka uthathe "Antabuse" icwecwe? Iingcali Guest zithi ingqalelo ichiza kufuneka ingamiselwa ukuba:
- glaucoma;
- neuritis le optic nemithambo eziviwayo;
- tuberculosis pulmonary;
- izifo sentliziyo semithambo (umz, post-iqhosha ithi, wavakalisa cardiosclerosis, yamafutha nobeempahla yobuchopho, isifo unesifo, kwemithambo aortic);
- polyneuritis nasiphi na imvelaphi;
- diabetes;
- emphysema, isifuba inyumoniya;
- thyrotoxicosis;
- ukugula ngengqondo, sokuwa kunye epileptiform syndrome;
- ithumba;
- hepatic kakhulu yaye ukusilela kwezintso;
- izifo hematopoiesis;
- exacerbation kwesifo isilonda Peptic;
- nokukhulelwa;
- hypersensitivity.
Kananjalo qaphela ukuba le echiza Izimo isihlobo:
- kweminyaka engama-60;
- imiphumo zestrowuku ezineempawu intsalela;
- isilonda Peptic (kuqukwa kuxolelwe);
- ngokwemvula a ngengqondo.
Drug "Antabuse": imiyalelo yokusebenzisa
Ipilisi ixabiso Anti-utywala ezidweliswe ekupheleni kweli nqaku. Kufuneka athathe embilinini ½ ngaphambili iqhawulwa iglasi yamanzi.
Ngokuqhelekileyo, amagqirha ukumisela 200-500 mg iziyobisi kanye okanye kabini ngemini. Emva kweentsuku 7, qiniseka ukuba bachithe uvavanyo disulfiram-utywala. Ngaxeshanye kunye ulwamkelo 500 mg yeziselo medicament nomonde 20-30 ml yevodka. Ukuba abasabela obuthathaka, ngoko ukunyusa ithamo kotywala ml-20.
Olu vavanyo iyaphindwa izihlandlo eziliqela. umdaniso kamva emiselweyo ulondolozo umthamo mg 200 imihla iminyaka 1-3.
ukusabela ezingalunganga
Tablets "Antabuse", apho amanqaku zinikiwe ngezantsi kunokubangela iziphumo ebezingalindelekanga kulandelayo:
- hepatitis, asthenia, metal incasa emlonyeni;
- obubonakala cutaneous, iinyawo polyneuritis;
- ukulahlekelwa inkumbulo, ukudumba kwengqondo, intloko ebuhlungu;
- iposi engabalulekanga, arrhythmias intliziyo;
- ukusilela yokuphefumla, ekuweni sentliziyo;
- neuritis optic, iimpahla thrombosis ebuchotsheni;
- kwengqondo, angina.
Medicament "Antabuse": Ukubuyekezwa amagqirha kunye nexabiso
Iindleko iipilisi anti-utywala malunga 450-600 engange (ngokuxhomekeke idosi kunye nemali pack ngalinye).
nangoko noogqirha amisele ichiza enjalo, walumkisa iingxaki ezinzulu ezingakhona isigulane kwisiqalo kuya kuthatha. Ngoko ke akuvumelekanga ngokungqongqo ukunyanga ngokwakho okanye imfihlelo evela isigulane.
Kufuneka kuqatshelwe ukuba iingcali ezininzi ziyavumelana ukuba amachiza asebenza ukuba gqiba njengokufuna utywala, akukho. Kwaye le ndlela ayikho unyango. It nje likhuthaza uyekelelo izinzile.
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