ZempiloAmalungiselelo

Metoprolol-ratiopharm

Metoprolol-ratiopharm zibandakanywa iqela amachiza asetyenziswa unyango lwezifo sentliziyo. Amayeza fanele ukuba iqela amayeza ibeta-blocker.

Metoprolol tablet ilifa iqinile, antiangialnym nesiphumo antiarrhythmic. Ichiza ithintela uphuhliso migraine.

Njengoko blocker ukukhetha beta, metoprolol-ratiopharm xa usebenzisa amathamo zonyango medium lineziphumo ezincinane izitho eziqulethe beta--adrenoceptors 2 (umsipha skeletal, injeke, emithanjeni neuropathy izihlunu agudileyo wesibeleko, yaye bronchi), kwaye kwakhona ekudleni ukutya. Ngoko ke amanyathelo atherogenic ezivakaliswe kumlinganiselo olufanayo xa usebenzisa propranolol. Xa kuthathwa ngeedosi ezinkulu Metoprolol-ratiopharm linamandla isiphumo uvimba kwi andrenoretseptory beta-1 beta-2.

Xa isicelo ngaphakathi iphawulwe ukufakwa epheleleyo (95%). Metoprolol-ratiopharm asasazwa ngokukhawuleza zomzimba, ingene nge njengomqobo placental, BBB.

Ichiza umzimba esibindini, le metabolites musa ukwenza igalelo ekhethekileyo umsebenzi beta-adrenoceptor ukuvimbela umlinganiswa.

Ichiza iboniswe lwegazi (zombini ngokuzimeleyo njengenxenye yonyango indibaniselwano kunye namanye amachiza umfutho), kweepesente intliziyo indalo esebenza kunye tachycardia. Yabela metoprolol kunye nesifo sentliziyo kobuchopho: iposi engabalulekanga (njengokuba nokuthintela eziziisekondari), angina (nokuthintela nokuhlutha). Iyeza eboniswe ekuthinteleni arrhythmias ventricular kunye tachycardia supraventricular, ngokunjalo migraine.

Le medicament asetyenziswe ngobunono izigulane seswekile sinwenwa, isifuba, lactic metabolic in sezintso (kwesibindi) ukusilela, thyrotoxicosis, myasthenia gravis, ukhwekhwe, occlusive isifo peripheral semithambo, ukukhulelwa, kunye nokuguga.

Metoprolol-ratiopharm. umyalelo

oyidlayo waqale lwegazi ngu-50 mg. Kwimeko okwenzeke yokungeneli unyango, ukuze zinongezele ku 100-200 mg okanye injongo ngakumbi ezinye amachiza umfutho. idosi yemihla ngemihla (ubuninzi) 200 mg.

Ichiza sithathwa ngomlomo, ndawonye namanzi, kanye ngosuku ngoko nangoko emva kwesidlo. Tablets akufuneki ukuhlafunwa.

Njengoko amanyathelo othintelo okuthintela yokuhlaselwa angina kokuqala idosi yemihla ngemihla ichiza-50 mg. Kwimeko ngempumelelo zaneleyo unyango ukuze zinongezele ku 100-200 mg okanye isabelo ezongezelelweyo antiangialnyh amanye amayeza. idosi iphezulu ngosuku - 200 mg.

Ukwenzela ukuthintela uhlaselo migraine ukuthatha iyeza ngosuku ka 100-200 mg.

Ukususela mg 50 ukuya 200 ichiza yayisalawulwa ukuphazamiseka ezisebenzayo kwentliziyo sikhatshwe yi tachycardia.

Xa zokuthintela (eziziisekondari) iposi engabalulekanga medicament ilawulwa ngendlela umthamo 200 mg ngosuku.

Xa insufficiency kwezintso, idosi ayidingi ukulungiswa. Kuxhomekeka kwimeko kwezonyango ukusilela hepatic Inokwenzeka isidingo esinjalo.

Ukuthatha iyeza iziganeko rhoqo ezingalunganga njengoko bradycardia, kuyithi abandayo yesiqephu asezantsi, hypotension intolerance (kuquka syncope), ukudinwa, isiyezi, ixhala, ukwanda ukucaphuka luvo, kwekhono ngokwesondo, isicaphucaphu, iintlungu esiswini, urhudo okanye ukuqhina, dyspnea on kuso.

Rhoxisa ichiza wavelisa ngokuthe ngcembe ngoxa kuncitshiswa esithathwa iiveki ezimbini. Kufuneka kuqatshelwe ukuba ukulahlwa usiko mali isekude noxinzelelo lwegazi, ukwanda lokuhlaselwa angina.

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