ZempiloAmalungiselelo

"Clonazepam": ncomo. "Clonazepam": imiyalelo ukusetyenziswa, imiphumela emibi

"Clonazepam" - iziyobisi antiepileptic leyo inxulumene avela benzodiazepine. Emva kokufumana i "clonazepam 'ukureyithwa eziseleyo iziyobisi ubukhulu becala HIV. Eli chiza relaxant kwezihlunu kunye neziphumo umthomalalisi, kodwa ibe okulalisa.

Ekwakhiweni, ifomu ukukhululwa "clonazepam" iziyobisi

Ichiza ifumaneka emacwecweni okubhalwe ezahlukeneyo amacandelo aphambili:

  • 0.5 mg. Ukongeza clonazepam, isakhiwo iquka monohydrate lactose. Ukuze izithako amacwecwe isebenza sodium carboxymethylstarch. "Clonazepam" Amaxwebhu aqulathe wemagniziyam stearate, awu. Nezincedisi nawo talc namazambane istatshi. Amacwecwe Umbala ngedayi E110 apha.
  • 2 mg. izithako olongezelelweyo abangabancedani - polysorbate 80, monohydrate lactose. Ukubunjwa langoku carboxymethylstarch sodium kesodiyam lauryl sulphate iziyobisi. talc, gelatin na izithako ozikhethelayo. Amacandelo Auxiliary and lilungu kwezinye izinto - wemagniziyam stearate, irayisi, itapile istatshi.

isenzo amayeza "clonazepam" iziyobisi

"Clonazepam" isiphumo ngxelo imbi kwinani elikhulu kwezakhiwo ezakha luvo central, ikakhulu abo ukuba ezinxulumene nemisebenzi ngokweemvakalelo. Isiphumo ichiza "clonazepam" umyalelo manual, ingxelo uboniswa njengoba sine, anxiolytic kunye thile (yokugqibela abangaxhalabisiyo wavakalisa). Le medicament kunciphisa kwezihlunu skeletal, kuthintela ukugula ngokubanzi convulsive. Kukho nempembelelo entle ekuhambeni kuhlaselo sokuwa (focal, ngokubanzi).

Pharmacokinetics

Ichiza ako phantse ngokupheleleyo ukusuka iphecana zesisu umntu ofakwe kakhulu izintso (metabolites), inxalenye minor (2%) ebonakala ingatshintshanga. Le nqubo ithatha isiqingatha ubomi iiyure eziyi-20 ukuya kuma-40. Le bioavailability sokulungiselela tapeworm yi-90%, ulwalamano kunye nonikezelo igazi - 85%, i ndzo iphezulu afikelela a kusho iiyure 2.5. Xa unyango "clonazepam" kwanangamacandelo alo ukungena ubisi lwebele.

Iimpawu zibonisa ukuba ukusetyenziswa kweziyobisi

"Clonazepam" macwecwe abafanelekileyo ukuba unyango izigulane yobudala ezahlukeneyo kunye sokuwa, kungakhathaliseki obubonakala:

  • ukuxhuzula inxenye (local, focal) nawuphi degree of abawayo
  • iimeko convulsive (indihlaziya, clonic);
  • nokuxutha izinto ezilula secondarily ngokubanzi;
  • ukungabikho Nedlac (Lennox-Gastaut syndrome);
  • zesifo myoclonic;
  • ukuxhuzula ukungabikho eqhelekileyo;
  • wokuqinisa-clonic ukuxhuzula imbonakaliso eziziprayimari nezizisekondari.

"Clonazepam" emiselweyo ukunciphisa kwezihlunu, zombini thile ubunzima kunye lengqondo ngexesha unyango.

Ukusetyenziswa kweziyobisi "clonazepam"

Umthamo ezifunekayo kumiselwa ngokusekelwe kwizinto ezininzi. Ngelo lokuqala unyango isebenzisa igcuntswana leyeza ekuthiwa "clonazepam" (0.5 mg), ngokuthe ngcembe ukutshintsha esithathwa de yifuna ifunyenwe. Ngelo xesha ngaphezulu idosi iphezulu kuyathintelwa. Njengoko ncomo, "clonazepam" ayikwazi ziphakame waphakamisa naxa unyango mfutshane ixesha elide. ukulahlwa usiko ichiza esongela uphuhliso i nokuhlutha sokuwa.

Ukwamkelwa for sokuwa:

  • Abadala. unyango lokuqala lwenziwa ngokusebenzisa hayi ngaphezulu kwe-1 mg iziyobisi. Ithamo ibalwa ngosuku, zibe-3 okanye 4 iingedosi, ekufuneka wenziwe rhoqo. Ngaphandle ukukwazi ukusebenzisa ichiza ngeedosi ngokulinganayo, elona "clonazepam" ethululwayo naphambi kokuba uye kulala. Ngokuqhelekileyo, ngendlela eyaneleyo imihla kuluhlu ka-4 ukuya kwi-8 mg iziyobisi. Ithamo yesondlo akufuneki ngaphezu kwama-20 mg (kuphunyezwa ngexesha kwiiveki 2-4 unyango). Xa ithamo olusebenzayo yemihla ngemihla, nto leyo evumela ukugcina imeko eqhelekileyo umzimba kumiselwa, uvunyelwe ukuba idosi enye ebusuku.
  • Abantwana (ngokobunzima ubuncinane 30 kg). Njengoko ncomo, "clonazepam" ekuqaleni eboniswe abantwana 0.5 mg ukumisela yedosi intsulungeko.

Reception kunye syndrome, sikhatshwa ziintlungu paroxysmal:

  • Abadala. Okokuqala, xa izigulane elawulwa 1-2 imini nomthamo (0.5 mg ngexesha ngalinye). izigulane ezininzi ezaneleyo ithamo enyangayo yi-1 mg / ngosuku. Emini ukusela ngaphezulu kwe-1 mg of "clonazepam" iziyobisi. Ukuphononongwa, Noko ke, zibonisa ukuba kwezinye iimeko, oogqirha kunokwandisa ithamo ku-4 mg. Kwiimeko ezinjalo, idosi ebegqwese zitshintshiwe (uluhlu - iintsuku ezi-3, mhlawumbi ukudibanisa 0.5 mg). Xa ufuna ukunciphisa ubuzaza nobuthongo ngexesha lasemini, ithamo libalwe yokwamkela ngexesha lasemini, ungakwazi kudla phambi lokulala.
  • Abantwana. Kuba izigulane abangengawo kweminyaka eyi-18, ekufumanekeni ichiza syndrome inokuba ingaphumeleli nezingakhuselekanga.

Ukuthintela naziphi na iingxaki, ichiza "clonazepam" reviews oogqirha bacebisa ukuthatha ngokungqongqo phezu izindululo ingcali okunyangayo.

Izimo ekufumaneni "clonazepam" iziyobisi

Iipilisi azisetyenziswa xa landa uvakalelo izinto apho zenziwe. Ichiza contraindicated kula ithi:

  • myasthenia gravis;
  • lomonakalo lokuqonda;
  • ukuzala, isikhuselo-lweehagu;
  • glaucoma (ukuvalwa);
  • izifo zemiphunga ukuba imvelaphi esembindini, kakhulu insufficiency sokuphefumla;
  • Heavy yhuu uxabane ukusilela hepatic;
  • ezabonakala elele syndrome;
  • ubuthi utywala;
  • ifomu abukhali porphyria.

Iziphumo ebezingalindelekanga "clonazepam" iziyobisi

Cinga iziphumo ebezingalindelekanga, esinokubangela "clonazepam". Ukusetyenziswa ichiza ukuze ezinxulumene ngayo ezibi. Kunokubangela ukuba silale, isicaphucaphu, ukuba nochuku. Ukuba uxabane yi umzimba womntu uyakhathala ngokukhawuleza, uye waba nolungelelwaniso kweentshukumo. Ukunciphisa isiphumo ngokubonakala of ziziphumo ebezingalindelekanga, kufuneka uqale ukusebenzisa igcuntswana leyeza, ngokwenyusa kancinane de kube kangangoko.

Yinto eyaziwayo ukuba ngexesha unyango "clonazepam" ithetha ulisebenzise waphula umthetho izindululo kungabangela libanda. Kwiimeko ezinjalo, kukho eyothusayo, nto leyo inokukhokelela nasekudaneni, badengeka, leyo kunokubangela isiqaqa. Phakathi kwezinye iimpawu - ukuwa semithambo, ukuphefumla kakuhle, ukozela. Kuyimfuneko lokuhlamba isisu (ngempumelelo ngoko nangoko emva kokudla iipilisi) ukuqhuba unyango olufanelekileyo. Kubalulekile ukuba esweni rhoqo utshintsho kakuhle kwizinto ezifana noxinzelelo lwegazi, ukubetha, ukuphefumla. Kwezinye iimeko, oku kufuna ukuphunyezwa umoya ngomatshini. Kukho esiphilisa - "Flyumazenil," kodwa akukho ezifanelekileyo zolawulo abaguli siphathwa "clonazepam" ixesha elide.

Akukho mfuneko ukudibanisa "clonazepam" kunye notywala. Ukuphonononga kuvumela ukuqinisekisa ukuba ukuhlanganiswa onjalo inokuba yingozi ebomini. Kukwasebenza kwanjalo kuyo zonke iziyobisi kusebenza kwinkqubo luvo, ziyibuyisela umsebenzi wayo.

Drug intsebenziswano "clonazepam" ukulungiselela

Ifuthe iyeza ukunyusa analgesics ezidakumbisayo, anticonvulsants. Isiphumo linye babonwe ngokudibanisa kunye lakhula, neuroleptics, barbiturates, nayo xa idibene kunye notywala kunye lunezinto ninganciphisi kwezihlunu skeletal. Impumelelo unyango lifinyele xa tapeworm nicotine.

Iindleko, ukubuyekeza ichiza "clonazepam"

Thenga "clonazepam" iipilisi eMoscow kungaba kuba 97-150 engange. (30-PC.). Ichiza iyasebenza sokuwa, ukuba zithotyelwe nengcebiso kagqirha. Xa ukuxhuzula atonic inokuba kweenyanga ezimbini, ubude unyango kwanele ngenxa yexesha elinje, uyakwazi ukukheta kunyango yesondlo. Ngamanye amaxesha kukho iziphumo ezingalindelekanga, kodwa ubukhulu becala kuphela kwisigaba sokuqala unyango, ngokufuthi ubuthathaka.

Xa ulwazi eziqulethe ncomo, "clonazepam" inqamla buncothulwe kwezihlunu kwanda malunga neeveki ezintathu. Amayeza amayeza xa umkhosi, uloyiko, IRR, nto leyo sikhatshwa uphaphazele. Ichiza kakuhle, isebenza ngokukhawuleza.

Izimvo "clonazepam" iboniswa njenge njengendlela elungileyo ukuba enze umsebenzi walo, kodwa kunokukhokelela yempilo enkenenkene (ubuthathaka, ukudinwa, njalo njalo. P.).

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