Zempilo, Amalungiselelo
"Bisoprolol": ncomo, imiyalelo esetyenziswa kunye analogue
Ngokutsho oogqirha, intliziyo yomntu - lelona candelo ibalulekileyo. Kungakhathaliseki ukuba yintoni imeko kunjalo, oku kuya kuxhomekeka kumgangatho wobomi kunye nexesha layo. Nayo nayiphi na umkhuhlane okanye izifo emathunjini abantu babuyelayo kwiikliniki rhoqo. Wonke umntu uyazi ukuba kunqabile kukhokelela ekufeni. Inxalenye isizathu apho umntu afe, ukuba isifo sentliziyo. Oosonzululwazi kunye cardiologists wadala ezininzi ngemithamo ukuba kuphela ukunceda ukwenza ubomi babantu, kodwa unako ubuncothule sifo. yaye lithetha "Bisoprolol" libhekisela kwiziyobisi ezinjalo. Ukuphonononga ezingeniswe amagqirha kwiijenali zonyango zibonisa ukuba izigulana isifo sentliziyo, wegqitha emva kwekhosi yonyango nalo eli chiza kuba lula kakhulu.
Main malunga kulungiselelwa "bisoprolol"
Eli chiza, nto leyo B-andenoblokiruyuschim ithetha. Kuye kudala isetyenziswa yezonyango, elileli: zentliziyo. Misa kuphela lwegazi, isifo sentliziyo, kodwa ukusilela intliziyo nezidubedube isingqi amayeza "bisoprolol 'intliziyo. Izimvo ezigulane zibonisa ukuba emva kweentsuku ezimbini ukuphelelwa ezilahlekileyo umoya, neentlungu entliziyweni.
A bit yomlando
Lo mbono lokukhupha iyeza efanayo wabonakala ngowe-1967. It wadalwa yi inkampani esebenza "Merck" (ukuba yinxalenye ngoko ke namhlanje liqela leenkampani "Astra"). Kwaba ngaloo nyaka okokuqala ngqa, oosonzululwazi baye bafumana into efana beta1-blocker. Ngaphezu koko, iintlobo zeHPV zingonobangela ezimbini receptors adrenergic sele ifunyenwe ngokusekelwe kwayo. Kuyinto ezifana B1-adrenoceptor kunye B2-adrenoceptor. Le medicament "Bisoprolol" libhekisela kwiqela blocker beta1-adrenergic uyakhetha. Bona uphawulwe uyakhetha kakhulu nezibekekileyo kwezinye izinto amandla.
Ukubunjwa ichiza "bisoprolol"
Ukuba sicinga amacandelo usemthethweni ichiza, oko kunokubonwa ukuba element engundoqo - iziyobisi yi bisoprolol fumarate ngokwayo. Iqulethe 5 iigrem iziyobisi zonke iipilisi "bisoprolol". Izimvo ezigulane zibonisa ukuba sele emva ukuthathwa lokuqala ichiza iphucula kakhulu zempilo. Akukho yeza na kwenziwa ngaphandle amalungu abancedisayo. Kwaye iziyobisi esebenzayo nayo iquka isodiyam croscarmellose okanye primeloza, povidone okanye polivinillirolidon srednemolekurny, starch prozhelatininy, lesilicon dioxide colloidal kunye talc encinane, microcrystalline kwincindi, lactose okanye ubisi iswekile kunye wemagniziyam stearate.
Uninzi imithi yayisoma egudileyo nencasa. Oku kusebenza ichiza "bisoprolol". Ukuphonononga zibonisa ukuba macwecwe angawokubhuda kakuhle, yaye akuyi kuhlala incasa krakra emlonyeni. Oku zonke enkosi amacandelo afana Macrogol (polyethylene ethers), titanium dioxide, Opadry 2. A iingqalutye umbala ezimnandi efunyanwa ngedayi ezisetyenzisiweyo - oxide yentsimbi (2).
Imiyalelo yokusebenzisa "bisoprolol" iziyobisi
Faka olu nyango iimfuno ezimiselwe kuphela ngugqirha. Kukho kusoloko nganye machiza iphakheji "bisoprolol" zikhombisa. Ukuphonononga zibonisa ukuba ngamanye amaxesha oogqirha bacebisa izigulane zabo izifundo elifuna ezahlukeneyo zonyango. Kuxhomekeke sifo, ubudala, iimpawu eziphilayo. Oku kudla Kucetyiswa ukuba basebenzise hayi ngaphezulu kwama-20 mg ngosuku. Oku iqhelekile omdala. Enye tablet idla 5 mg. Kufuneka ukuba zingahlafunwa kwaye kufuneka wabaginya namanzi amaninzi. Ezo zincomo zibandakanya ukuba ichiza "bisoprolol" umyalelo manual. Izimvo kwesokunxele abantu abaye basebenzisa oko, ubonise ukuba ikhondo emva wadlulisela impilo unyango iba ngcono kakhulu.
Ukuba isigulane ixabisa uxilongo "lwegazi" okanye "isifo sentliziyo", kuyimfuneko ukusebenzisa iipilisi 2 ngosuku, ngokuqhelekileyo kusasa nangokuhlwa. Inxaxheba kwinqanaba lokuqala idosi unyango kube incinane - 5 mg kuphela ngosuku okanye tablet nye. Ngokuzimela ukudlula eqhelekileyo kuyo nayiphi na imeko engenakwenzeka. Ukuba iyeza swi nga pfuna, kufuneka kuqala udibane nogqirha wakho kwaye senze yeziphakamiso yayo. Iingcali kokuba ukumisela le amayeza, khangela umsebenzi namanye amaqumrhu kunye ingqalelo ekhethekileyo ihlawulwe nokubetha kwentliziyo. Phambi kokuthatha iipilisi kwisigulana kwaye kufuneka ukukhangela izinga intliziyo yakho.
Izimo
Nayiphi medicament kwabantu zizifo ezahlukahlukeneyo kunokubangela iziphumo ebezingalindelekanga ezingathandekiyo. Oku kukwasebenza "bisoprolol" iziyobisi. Iimpawu zibonisa ukuba ukusetyenziswa sele phakheji ngamnye. Le ncwadana ithi ukuba akukho mfuneko yokuba oku iyeza isicelo yokothuka, bradycardia (izinga intliziyo ukuba ibetha ngaphantsi kwama-50 imiz nganye.). Awukwazi ukusebenzisa oko, naphantsi kwafa atriovenkulyarnoy izidanga-2 no-3, kwaye ukuba kukho syndrome of uju of sinus node kwaye ukuba hypotension libizwe.
Kwakhona, ichiza kuyimfuneko ukuba ngaphandle abantu hypersensitivity okanye bewenza bronchospasm. Ukuba izigulane ziye phambili ibakala ukuphazamiseka peripheral yokujikeleza, iyeza nalo ayifanelekile. Awukwazi ukusebenzisa amayeza "bisoprolol" (ixabiso layo yi-avareji engange-30.) Yaye xa isetyenziswe Mao inhibitor (kodwa akukho inhibitor Mao-B).
Iintsilelo lolwamkelo esikolweni "Bisoprolol" ukulungiselela
Faka isiyobisi esebenzayo kufuneka ngenyameko abantu abaye izifo ezifana neswekile sinwenwa, hypoglycemia, lactic metabolic, thyrotoxicosis, atrio-ventricular block 1 vazospasmaticheskaya isidanga angina. Kwakhona Awukwazi ukusebenzisa eli chiza kwizigulana bangekhoyo ukutya engqongqo, yaye abo baye benza ikhosi efana therapy nemithi.
Xa isifo enjalo, njengoko ukusilela intliziyo ayikwazi ingasetyenziswa ngexesha exacerbation iziyobisi "Bisoprolol". Ukuphonononga zibonisa ukuba le meko ukusetyenziswa kweziyobisi kungaba kubi impilo. Kwakhona lo uphethwe kufuneka usebenzise eli yeza ukuba ireyithi intliziyo ibetha ngaphantsi kwe-60 ngomzuzu. Kwakhona kubhaliwe contraindicated kwaye kunciphise uxinzelelo lwegazi iSystolic, ingakumbi xa lingaphantsi kwe-100 mm HG.
Medicine "bisoprolol" kunye nokukhulelwa
Le ichiza kuyo nayiphi na imeko ingenakusetyenziswa kulophulo abafazi abakhulelweyo kunye phindeke. Kukho iimeko, xa kuyimfuneko ukuba aphilise isigulane kunye ngokuzala, kodwa kufuneka asiyeki ukusebenza xa, phambi kokuzalwa imalunga 72 iiyure. Ukuba oku akwenzeki, ngoko usana kufuneka igcinwe phantsi kweliso oogqirha ukusuka kwimizuzu yokuqala yokuzalwa. Lo mntwana, emva eli chiza inokuphuhlisa hypoglycemia, kwaye ukubonakalisa sifo sele kwiintsuku ezintathu zokuqala.
imiphumela emibi
iziphumo ezibi babe phantse zonke iziyobisi. Medicament "bisoprolol" inokuyichaphazela luvo. Oku kubonakala ukudinwa, isiyezi, intloko ebuhlungu rhoqo, zokulala. Kukudakumba kwenzeke kwiimeko ezinqabileyo, nemibono. Kodwa oku konke kwenzeka ngendlela elula, yaye emva kweeveki-1 okanye ezi-2 emva kokuba unyango kwenzeka.
ziphumo bezingalindelekanga kungahle kuchaphazele amalungu yombono ngohlobo conjunctivitis okanye anciphise ukukrazula. enqabile nje uphelelwa ngumphefumlo Inokwenzeka, kodwa oko kwenziwe ngabantu abathanda bronchospasm. Ngamanye amaxesha oko ngazo yaphula phecana zesisu. Okungakanani isicaphucaphu okanye isifo sorhudo, amahlaba luncinane esiswini. Kodwa izifo lolu kwiintsuku ezimbalwa kudlule.
analogs
Ngu analogue beziyobisi "bisoprolol" ziquka indlela lekartsvennye:
- "Concor".
- "Biprol".
- "Niperten".
- "Bisogamma".
- "bisoprolol-UPramila."
- "bisoprolol-ukuziqeqesha" kunye nabanye.
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