Lithetha othi "Tranexamic acid" yi ichiza antifibrinolytic, inyathelo anti-ukudumba kwaye antiallergic, kwakunye endibuthethileyo ukusebenza hemostatic xa bleedings enxulumene ne ukwanda fibrinolysis. Xa ingundoqo ichiza na inhibition of plasminogen isilumeki kunye plasmin inhibition ye ukuyilwa peptides esebenzayo kunye kinins ababandakanyeka ngqo reactions ukudumba kunye negazi. Ukongeza, isixhobo ezifana "Tranexamic acid", alongezi kakhulu ixesha thrombin. Ngokumalunga iimpawu pharmacokinetics beziyobisi anti-fibrinolytic emva kokungenisa kokuba ako malunga ne30-50% of umthamo wayo ekuqaleni, le boxinzelelo ephezulu plasma kuphawula ikhulu - imizuzu ikhulu elinamanci asibhozo emva kokuba usebenzise amachiza. ukusebenza Antifibrinolytic zomzimba Bagciniwe elinesihlanu - iiyure elinesixhenxe, plasma - iiyure ezisixhenxe okanye ezisibhozo emva ulawulo ichiza "Tranexamic acid". Ixabiso le sixhobo imalunga 1300 engange, kwaye ukuyithenga phantse yonke ekhemisti.
isiyobisi Antifibrinolytic iveliswa ngokohlobo amacwecwe ezingamakhulu amabini anamashumi mahlanu okanye anamakhulu mahlanu mlligrams, njengoko isisombululo ukuba isitofu, kwakunye isisombululo elungiselelwe ulawulo ngomlomo. Zonke iifom idosi ngasentla kakuhle ifanele ukuba unyango kunye nothintelo ukopha, wamqumbisa ukwanda fibrinolysis lulonke. Umzekelo, i-arhente kaninzi elawulwa, apha ochazwa ngokuba "Tranexamic acid 'xa yamathumba amabi, ze endlaleni okanye nepancreas, wegazi, ungenelelo zotyando phezu amalungu esifubeni, kunye izifo zesibindi. ukususwa Manual of ngumkhaya kunye Kukudandatheka legazi nazo zifakwe kuluhlu lwe ezibonisa ukuya kuyo. Ukongeza, ukusetyenziswa kweziyobisi "Tranexamic acid 'kufuneka of haematuria, angioedema, dermatitis negazi, nangokhwekhwe, ityhefu kunye neziyobisi irhashalala, ezindlwini. Ukongeza, eli chiza iboniswe ngenxa pharyngitis esebenzayo, laryngitis, tonsils, stomatitis, ukuthetha kwam ngeempumlo, zesibeleko kunye isisu ukopha, izinyo xa izigulane ukuba unesifo ukopha diathesis. Njengoko kakuhle ukuba isixhobo ezifana "Tranexamic acid ', kunye ngenyanga, ngaphandle enkulu.
Njengoko isicelo namayeza wemithi, kwimeko nganye ukuba ibekwe ngamnye, esekelwe kwimeko banikwa lwezonyango. Noko ke, njengokuba umthetho, ngexesha uvumelekile ukuba zaba ngaphezulu kwe 1-1.5 grams. Kulo mzekelo, ukusetyenziswa ubuninzi kukuba izihlandlo ezibini ukuya kwezine ngosuku, kunye nobude unyango - ukusuka kwiintsuku ezintathu ukuya elinesihlanu. ithamo Single lolawulo efakwa yi 10-15 mg / kg.
Eyona Izimo eziphambili ukuba basisebenzise esi sixhobo kukho iimeko ezifana legazi subarachnoid, thromboembolism, ukusilela kwezintso, nokuphazamiseka umbala imbono, yaye zinzulu vein thrombosis. Ukongeza, kufuneka asebenzise eli amayeza xa kukho hypersensitivity okanye yokukhulelwa. iziphumo ebezingalindelekanga ezinxulunyaniswa ne lokuthathwa arhente anti-fibrinolytic, ibonakaliswe njengokuba nesiyezi, nobuthongo, hypotension, tachycardia, ukutyhafa, kunye neentlungu esifubeni.