Zempilo, Amalungiselelo
"Motonium": imiyalelo, real
Phantsi nokugabha kubonisa dubulo (reflex) iziqulatho esiswini ngomlomo. Ngokuqhelekileyo, inkqubo enjalo landulelwa isicaphucaphu kunye ligwinya ubhalo ngengozi, secretion oluncediswayo iinyembezi, ematheni nokuphefumla ngokukhawuleza.
Kunye iintsalela ukutya, ijusi esiswini, yencindi, duct nezinye ubumdaka, indoda ejaculates kunye nezondlo. Oku kunokubangela emzimbeni kunye electrolyte ukungalingani. Ngoko ke, xa nokugabha eyomeleleyo kunye rhoqo, qiniseka ukuba inani lamanyathelo ukuba uya kusindisa zonke izimbiwa kunye nezinye izinto emzimbeni womntu.
Enye antiemetics kakhulu ethandwayo "Motonium". Imiyalelo yokusebenzisa, kwiipropati zokwenene kunye Izimo beziyobisi zidweliswe ngezantsi.
Ukubunjwa ichiza, zayo imilo, ukupakisha kunye nenkcazo
Ziziphi ifomu ukhulula ichiza "Motonium"? Guide ingxelo ukuba le mveliso yenziwa ngokohlobo ngeenxa kunye neepilisi bhanya-camera emhlophe. isithako yabo esebenzayo uba domperidone. Kwakhona zibandakanyiwe medicament: lactose, microcrystalline kwincindi, glycerol, umbona starch, nemagnesium stearate kunye ezisezantsi ezinto povidone weight. Ngokubhekiselele iveze inwebu, ukuba iqulathe hydroxypropylmethylcellulose kunye polyethylene ethers 6000.
Thenga iipilisi "Motonium" (ngawo bamiswe, siza kukuxelela ngezantsi) banokuba namadyungudyungu okanye iinkonkxa zeplastiki, ezipakishwe kwiibhokisi kwikhadibhodi.
Isenzo beziyobisi
iziyobisi "Motonium" Zisebenza njani? Imiyalelo isicelo ibonisa ukuba yindlela ukwandisa ixesha izishunqulelo peristaltic kwi duodenum kunye antrum esiswini. Ngaphezu koko, oko ibalekisa kakhulu yokulahla esiswini (ngexesha deceleration yenkqubo), ishenxisa imvakalelo isicaphucaphu nokugabha, kwakunye esophageal uyanda ithoni sphincter (ngaphantsi).
Yintoni na iziyobisi ephawulekayo "Motonium"? Ukuphonononga zibonisa ukuba ikhuthaza ukukhutshwa prolactin ukusuka ingqondo yebhinqa. ukusebenza kwayo anti-emetic kubangelwa impembelelo peripheral okanye gastrokinetic kunye kwingcinezelo receptors dopamine ibekwe kwindawo chemoreceptor adubule.
Kufuneka uqaphele ukuba domperidone alunasiphumo kwi secretion yejusi esiswini.
features kinetic
Yintoni Lubalasele kinetics beziyobisi njenge "Motonium"? Imiyalelo yokusebenzisa okufunwayo emva ezithatha ichiza, yena wendele kunokuba ngokukhawuleza.
Eli chiza bioavailability ephantsi (malunga ne-15%). Its lamanani igazi eliyincopho waphawula emva kwemizuzu engama-60.
Ukuncipha juice iasidi esiswini kunciphisa inkqubo ukufunxeka domperidone. Akazange ukungena umqobo igazi-ingqondo, ngoko ukusetyenziswa kwayo kunqabile kakhulu kunye neziphumo ebezingalindelekanga.
Le medicament "Motonium", imiyalelo zokusetyenziswa oboniswe apha ngezantsi, isasazwa kakuhle emzimbeni. Noko ke, ingqalelo yayo ingqondo ayinamsebenzi. Ukubambana kulungiselelo iiproteni plasma 91-92%.
Ngokubanzi umzimba esibindini na ekucaca ukuba ichiza kunye neendonga emathunjini. Its nesiqingatha sexesha-ubomi iiyure ezili-9, kwaye ukusilela kwezintso (ichazwe) kwisithuba ilandelayo elide.
Wabonisa kidney amayeza kwaye amathumbu.
Ubungqina obubonakalayo buxela ukuba abafumana iipilisi amayeza
Kwezinye iimeko, ukulungiswa nomonde "Motonium" linokukwenziwa? Izimvo oogqirha bathi ukuba iyeza lisetyenziswa entsonkothileyo kweempawu dyspeptic ezinxulumene reflux esiswini okanye esophageal, kudinga release esiswini okanye esophagitis. Ngenxa yoko, i-arhente isifundo isetyenziswa flatulence, imvakalelo ukuzala kwi epigastrium, uza ukuqunjelwa, belching, iintlungu esiswini eliphezulu, yaye heartburn ngaphandle ezikhupha (okanye, icala, kunye reflux) kwiziqulatho isisu emva emlonyeni.
Kwenye into kunceda iziyobisi "Motonium"? Imiyalelo yokusebenzisa ingxelo yokuba eli ukulungiselela ishenxisa imvakalelo isicaphucaphu, ukugabha, ithintela uphuhliso zohlobo ephilayo, ezosulelayo, kwaye esebenza, kwakunye okubangelwa radiotherapy, ukutya disorder, unyango ngamachiza kunye ulwamkelo agonists dopamine (umz: "Bromocriptine" okanye "Levodopa").
Izimo ukuba zifumana inkxaso-mali
Eli chiza ngononophelo Kucetyiswa ukuba abantu insufficiency hepatic okanye sezintso. Ukongeza, ukuba ungamiselwanga ukuba nesisu okanye ukopha isisu, hypersensitivity, kwesisu perforation, okanye esiswini isithintelo ngoomatshini isisu, kwakunye nobukho prolactinoma naphantsi kwiminyaka emihlanu.
Drug "Motonium": imiyalelo yokusebenzisa
Thatha le mali kufuneka ibe ngaphakathi imizuzu 20-35 phambi izidlo. Le umthamo ichiza kuxhomekeke imeko yesigulane.
Xa abantwana ukuqunjelwa ezingapheliyo kweminyaka emihlanu medicament elawulwa 2.5 mg / 10 kg ubunzima bomzimba kathathu ngemini. Kwiimeko kaxakeka ichiza athathwe naphambi lokulala. Njengoko abantu abadala, baya kumisela-10 mg beziyobisi (okt 1 tablet) kathathu ngemini kunye, xa kukho imfuneko - nje kokuba lokulala.
Ukuba kuyimfuneko, idosi elikhankanyiweyo angandiswa kabini.
In acute kunye subacute ithi (isicaphucaphu nokugabha) kwizigulane abadala zilawulwa 20 mg medicament (ngamanye tablets 2) kane ngemini, naphambi lokulala. Kids ukusuka kwiminyaka emihlanu esi sixhobo Kucetyiswa ukuba athathe 5 mg / 10 kg ubunzima bomzimba kathathu ngemini kunye ebusuku.
imiphumela emibi
Izincomo antiemetic azifane kubangela ngayo ezibi. Kukho amatyala amahlaba ezidlulayo isisu, kunye nezigulo extrapyramidal abantwana kunye nabantu nokonyuka permeability le BBB.
Ukongezelela, izigulane abafumana eli chiza lisenokuba negazi ezifana urticaria kunye irhashalala. Ngamanye amaxesha iziyobisi esebenzayo ebangela hyperprolactinemia (gynecomastia kunye galactorrhea).
Libanda kabi
Ziziphi iimpawu kwenzeka xa uthatha ngeedosi eziphezulu le mali? Iingcali zithi eli chiza kungabangela ukozela, nokudideka kunye abasabela extrapyramidal, ingakumbi ebantwaneni.
Kuba unyango kweemeko ezinjalo ixhoba isebenze wamalahle antihistamines. Xa antiparkinsonian kunye anticholinergics ukuba ekucetyiswa isahlakalo extrapyramidal reactions nomonde.
Intsebenziswano kunye nezinye iindlela
amayeza Anticholinergic yokungenelela ifuthe domperidone.
Sodium yesoda, "cimetidine" kunye nezinye protivosekretornye kunye asidi ukunciphisa bioavailability beziyobisi.
Antibiotics ngoweqela of macrolides, iziyobisi nokubola azole, "Nefazodone" kunye HIV protease inhibitors domperidone ukwandisa xiyimiso egazini.
Ukusetyenziswa in abasetyhini abakhulelweyo kunye phindeke
Drug "Motonium" inokusetyenziswa senyanga yokuqala yokukhulelwa, kodwa kuphela ezibonisa ezikhethekileyo.
Le domperidone ubisi lwebele boxinzelelo izihlandlo ezine kunonyaka plasma. Iingcali abazi nokuba nomphumela domperidone ezingentle bawo kwi kubelekwa. Ngoko ke, ibele kufuneka kupheliswa xa efumana iipilisi.
izincomo ezithile
Abantu abane insufficiency kakhulu kwezintso, iziyobisi isiqingatha-ubomi lanyuka ukusuka 9:00 20 Noko ke, uyazikhomba ichiza egazini usezantsi kakhulu kubantu abasempilweni.
Ngenxa yokuba eli chiza kwazona yi izintso ngezixa ezincinane, ukulungiswa kwayo iyunithi esithathwa xa izigulane lomonakalo sezintso ingafuneki. iyeza yedosi kunjalo ephindiwyo ubuninzi wayo kufuneka linciphiswe ukuze amaxesha amabini ngosuku (kuxhomekeke iqondo yokusilela).
Ulawulo Chronic nemithi, izigulane kufuneka abe phantsi kweliso rhoqo.
ixesha Ukugcinwa kunye nemiqathango nokuvalelwa
amayeza kujongwa kufuneka igcinwe kwindawo eyomileyo, ekhuselweyo ekukhanyeni kwaye zikhuselekile kubantwana abancinane. lobushushu yokugcina kufuneka abe ngaphezulu ko-25.
Ubomi lokugcinwa kwezinto ichiza iinyanga ezingama-24. Musa ukuthatha iipilisi emva kokuphela kwexesha elikhankanywe ekwibhokisi.
Drug "Motonium": ukubuyekeza isiguli
Malunga ingqalelo kuthetha kukho ncomo baninzi kangaka. Amaninzi, ukuba HIV. Abasebenzisi bathi eli chiza kakhulu ngempumelelo ekunciphiseni ukugabha kunye ishenxisa nokuziva isicaphucaphu. Ngaphezu koko, iziyobisi esebenzayo lidla kusetyenziselwa ukuzinciphisa iimpawu dyspeptic.
Ukongeza umsebenzi omkhulu, yemfaneleko eli chiza ziquka nokusilela Izimo ezinzulu nokufumaneka. Kufuneka kuqatshelwe ukuba ichiza "Motonium" phantse zange kunokubangela iziphumo ezingalindelekanga, kuqukwa abantwana abadala ngaphezu kweminyaka emi-5 ubudala.
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