Zempilo, Amalungiselelo
Izoptin: imiyalelo yokusebenzisa
Xa izigulane lwegazi ubeke izoptin. Imiyalelo zokusetyenziswa ichiza malunga ezibonisa, iziphumo ebezingalindelekanga kunye Izimo.
Ukongeza unyango nomfutho izoptin into esebenzayo i verapamil, zinayo angina kunye tachyarrhythmia. Phakathi kwezinye izinto, le alginates iziyobisi kunye polysaccharides ezivela ulwelwe (brown), ezisetyenziswa isiseko ezibonakalayo ukuze matrix hydrocolloid. Ukuba uthatha izoptin (imiyalelo ukusetyenziswa ngokucacileyo ibonisa kuyo) ngosuku kanye, isiphumo yayo kwezonyango kuhlala njalo elide. Oku iibhloko ichiza calcium channels, yehlise ukuxhathisa semithambo, ngoxa ukwandisa nezihlandlo kwamathumbu intliziyo. Ukongeza, verapamil kunye nokusetyenziswa rhoqo engaphenduli ukuphuhlisa arrhythmias sehlise e kwentliziyo inkanuko kwezihlunu.
Ukuba ugqirha uye wamisela izoptin, usuku emva kokuqaliswa ichiza isigulane kunciphisa uxinzelelo, yaye esi siphumo igcinwa, ukuba isigulane iyaqhubeka unyango lodweliso olucetywayo, ugqirha. Ngapha koko, uhlobo oluthile kunamandla ivumela ngokuqhubekayo, ukukhululwa phantse kumgama owazisayo eyona nto ebonakalayo ichiza, eqinisekisa ulondolozo umgangatho ichiza plasma.
Izoptin ako, lo myalelo ichanekile, emathunjini amancinci phantse ngokupheleleyo (90-93% degree of ukufunxeka). Ukuba ukuba bazithathe kanye ichiza, isiqingatha-umphefumlo wayo uya kuba iiyure 3-7. Ukuba indlela efanayo inde, kweli thuba iza kuba amaxesha ngaphezulu amabini okanye amathathu. Ukuboniswa izoptin, yemiyalezo zichanekile, ingakumbi inkqubo wokuchama, kwaye endleni yenani lilonke yayo-16%.
Ekubeni isithako esebenzayo yenziwe lula uleyisayo ngumkhaya, izoptin ngexesha lokukhulelwa hayi kuboniswa. Izoptin umi amasi kanina, kodwa amasi xi ayinamsebenzi, ngoko ke umntwana yena akanayo imiphumo imithi. Kodwa iingcali ingekabinazo singacebisi ukuthatha phakathi zisanyisa.
Emiselweyo ichiza becala ezi zifo zilandelayo:
- ukukhanya kunye nomyinge degree of lwegazi (monotherapy eyabelwe);
- degree kakhulu nomfutho (ezintsonkothileyo eyabelwe kunye nezinye iziyobisi - womchamo njl).
Kwakhona eli izoptin, imiyalelo zokusetyenziswa uzicacisa sebenzisa njenge arhente othintelo ukuba sifuba angina (kubandakanywa Pintsmetala) kunye tachyarrhythmias supraventricular.
Umthamo nayiphi na amatyala ikhethiwe ngqongqo ngabanye, kuba eli chiza Izimo. Umzekelo, mayingabi sakhululwa yabelwe abo basenokuba ukothuka cardiogenic okanye kwisigaba nokoyika iposi engabalulekanga nzima bradycardia, kuphazamisane ventricular ekhohlo, phantsi kwegazi. Ezingavumelekanga isidanga ukusetyenziswa isoptin kwafa AV II-III kunye sinoatrial. Ubulumko kufuna amayeza ngexa lokukhulelwa.
Phakathi iziphumo ebezingalindelekanga bradycardia, sinus, isicaphucaphu, hypotension, uvalo, intloko ebuhlungu, ukuqhina, paresthesia. Ekubeni eli chiza kunokubangela ukuphakuzela, isiyezi, ukudinwa, izenzo silale, ulwamkelo yayo ayinqweneleki xa uqhuba izithuthi. Ngexesha ukusetyenziswa isoptin asikwazi ukuthatha utywala.
Ukuvelisa izoptin azipilisi kunye mg 240 ukuya 120.
Olu nyango emiselweyo, njengesiqhelo, kwi idosi ilandelayo: ngosuku kanye okanye kabini, okanye ngaphambi kokuba isidlo okanye ngoko nangoko emva kokuba. Ngaloo non-absorbable tablet isoptin hayi zingahlafunwa kwaye wahlamba phantsi ngamanzi (a ubuninzi elincinane). Unyango nge verapamil (Isoptin) uxinzelelo lwegazi oluphezulu kuphela kwenziwe phantsi kweliso elibukhali likagqirha. Ngokubanzi ukuqala unyango nocingo mnye. Ukuba ufuna ukwandisa ukunciphisa of uxinzelelo oluphezulu lwegazi, ugqirha umisela poltabletki yokwamkela ngosuku (kusasa), ekupheleni kweveki yesibini ezikhokelela ukuya umthamo we 1-1.5. Emva kweeveki ezimbini, idosi inganyuswa ukuba amacwecwe amabini, kodwa ke kungekho ngaphezulu. Apho wesibini osuswe ngokuhlwa ukuze ixesha phakathi amathamo iiyure ezili-12.
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