Zempilo, Amalungiselelo
"Keppra" - ncomo. Anticonvulsants. Inkcazelo yokulungiselela, imfundiso
Sokuwa - sisifo yeqhelekileyo imisebenzi ezalanayo kwiqela neuropsychiatric. Le izigulo ezingapheliyo kwaye ayikwazi ngokupheleleyo unyangiwe kuyo. Isigulane unokuziva ocoliweyo ixesha elide. Xa ixesha nokuhlutha zizitye, nto leyo idala umngcipheko ubomi isigulane. Ukuze kuthintelwe ukuqhubela phambili sokuxhuzula, amayeza eyahlukeneyo asetyenziswa. iziyobisi Popular ebizwa "Keppra". Uhlaziya Iingcali ngako emihle.
ifomu Release komsindo
Ichiza ifumaneka azipilisi kunye isisombululo ukuba zisetyenziswe ngaphakathi. Amayeza bobabo kwiqela anticonvulsant. Icandelo engundoqo esebenzayo izenzo levetiracetam dihydrochloride. Njengoko excipients kusetyenziswa isodiyam croscarmellose, lesilicon dioxide, macrogol, wemagniziyam stearate. Le isisombululo Ukongezelela kusetyenziswa amacandelo ezifana sodium acetate trihydrate, isodiyam hayidroksayidi, kwaye acetic acid.
Pharmacokinetics
Emva kokungenisa "Keppra" (tablets) bathi bafakwe ngokupheleleyo iphecana zesisu. Adsorption lwento. Uyondelelwano lwee- icandelo ephambili plasma kube lula kwangaphambili ukusuka idosi ukuba isigulane sifumana. Le bioavailability beziyobisi yi-100%.
Xi iziyobisi liphezulu egazini bafikelela nesiqingatha seyure emva kokungenisa. Isiphumo therapeutic ukuze kubonwe kwiintsuku nje ezimbalwa phantsi imeko tablet kabini ngemini. "Keppra" isisombululo isebenza kakhulu ngokukhawuleza. Iziphumo zokuqala isigulane uyalibona Kusuku olulandelayo emva kokuqalisa unyango.
ubungqina
Njengoko monotherapy ezisetyenziswa yonke iziyobisi "Keppra". Ukuphonononga kubonisa ukuba unyango kuba neziphumo ezihle. Ngoko ke, ukusetyenziswa nezinye iziyobisi ayikho imfuneko. Ichiza uya kunyanzeliswa uxhuzula nanonelela abadala kunye nabantwana abangaphezu kweminyaka-4 ubudala kunye sokuwa. Xa ngokubonakala amayeza nokuhlutha mioklinicheskih nabo anikwe izigulane ezindala ngaphezu kweminyaka 12.
Le medicament ezingabantwana isetyenziswe ngobulumko. Nefuthe elibi kwizigulana abaselula ngaphambili iye waphawula. Nangona kunjalo, iingcali zithi abantwana siphathwa, inkumbulo ezahlukeneyo embi, kunciphisa kakhulu umnqweno ukufunda. Drug "Depakine Keppra" lisetyenziswa kuphela xa kwezinye, ii-arhente ezininzi engashiyi musa ukunika iziphumo ezidibanisayo.
Izimo
Kuye yayo Izimo iziyobisi "Keppra". Imiyalelo zokusetyenziswa ibonisa ukuba iziyobisi ifomu ipilisi ayikwazi anikwe izigulane ngaphantsi kweminyaka-4 ubudala. Kuba abantwana oko ukulungiselela olufanelekileyo ngakumbi njengesisombululo okanye isiraphu. Kodwa kule fomu oko kuthetha abantwana ongaphathiswanga ngenyanga yokuqala yobomi. Kukho zingasetyenziswa iziguli amayeza kuye kukho lunyhasho nokunganyamezelwa fructose. Ukungaphumeleli ukwenza oku kunokukhokelela nemiphumela emibi kakhulu.
Akunyanzelekanga amachiza abantu ukusilela kakhulu kwezintso kunye hepatic. izigulane abadala (kweminyaka engama-65) ichiza isetyenziswe ngobulumko. Unyango kwenzeka kwindawo yonyango phantsi kweliso gqirha.
oyi
Ukuba ufuna ukuba uyeke ukuthatha anticonvulsant, oku kufuneka kwenziwe kancinci. kumiwe ngokukhawuleza ukusetyenziswa amacwecwe okanye isiraphu engabangela ukuqala i nokuhlutha sokuwa. iziyobisi ebonakalayo chu irhoxisiwe.
Izigulane kufuneka wezintso kwaye zesibindi izifo, phambi kokuba unyango Kucetyiswa ukuba bangenele uphando olunzulu eziphilayo. Oku kuza kutyhila Izimo kunokwenzeka. Ichiza anticonvulsant kungaba nefuthe elibi function kwezintso. Kwezinye iimeko, kusenokufuneka ukulungiswa balawule.
balawule
amayeza "Keppra" ithathwa kabini ngemini. Kwimeko monotherapy kubaguli kweminyaka engama-ezilishumi elinesithandathu iziyobisi elawulwa ngohlobo amacwecwe. Ithamo yokuqala 500 mg ngosuku. Le ummiselo sahlulwe amathamo amabini ka-250 mg. Emva kwexesha elithile, idosi kufuneka kwandiswa ukuya ku-1000 mg ngosuku. Izinga eliphezulu ayikwazi ngaphezu 3000 mg.
Xa unyango entsonkothileyo abantwana abangaphezu 1 nyanga linokukwenziwa ukuba ichiza ngohlobo isiraphu. Umthamo uzimisele ngokusekelwe ubunzima bomzimba nomonde kwaye 7 mg 1 kg ubunzima nganye. Ukuba umntwana ubunzima isiyobisi eqhelekileyo, kwiveki enye idosi kufuneka kwandiswa ukuya ku-21 mg nganye 1 kg ubunzima. Unyango abantwana abancinane ngaphezu kweminyaka emi-3 kufuneka uthathe indawo ngqo phantsi kwiziko lonyango phantsi kweliso wabantwana. Esithathwa abantwana abanobunzima ngaphezu kwama-50 kg iyafana nje abadala (500 mg ngemihla).
Kuhle ukukhumbula ukuba ichiza "Keppra 500" kwazona yi nezintso. Ngenxa yoko, xa izigulane kuba kukutenxa ethile kulo mzimba, kusenokufuneka ukulungiswa idosi. Izinga mihla iya kuba ngaphantsi kancinane kunye nonyango lwabantu abadala ngaphezu kweminyaka engama-65.
libanda
Ngamana ukuphuhlisa iziphumo ebezingalindelekanga ukuba kudliwe izixa kakhulu iipilisi "Keppra". Ukuphonononga zibonisa ukuba iimpawu yokuqala libanda, kuba ukozela, isiyezi, isicaphucaphu, ixhala, ukudakumba lokuqonda. Ebusuku isiguli kube ubuthongo waphazamiseka, kuvela amabi.
imiphumela emibi
Iimpawu ezingemnandi zinokuvela xa usebenzisa idosi echanekileyo beziyobisi, "Keppra". Levetiracetam kwi sigaba sokuqala unyango kunokubangela ukozela ngokugqithiseleyo. Esi simo okwethutyana kwaye ayifuni ukupheliswa unyango. Isiguli nazo iimpawu ezifana yintloko, ukulungelelana kakuhle, kunciphise ingqondo, memory sokunciphisa.
Kwinkqubo okucola ukwehlelwa ziziphumo ebezingalindelekanga ezifana norhudo, ubucaphucaphu, ukugabha, ukungabi namdla. Kwezinye iimeko, ukuphuhlisa anorexia. Izigulane bayala ukutya maxa onke. Unyango kulo mzekelo kufuneka kwenzeka kuphela phantsi kweliso zonyango esibhedlele.
ulawulo Chronic yokulungiselela "Keppra" ziziphumo ebezingalindelekanga nga ha kombisa nokuxubana dermatological. Le ukurhawuzelela, ukuba bomvu, bechuba, amaqhakuvana amancinane. Kusenokubakho ongaboniyo. Isigqibo lokuphelisa ulwamkelo iipilisi okanye isisombululo kuthatha specialist. Kwezinye iimeko kwanele ukuba ukunyenyisa esithathwa ukuya ngokubonakala reactions ezibi lihlile.
imithi
Eyona nto ephambili esebenzayo modem kunye anticonvulsant. Ngoko ke, ichiza "Keppra" ukuze ziqukwe kunyango entsokothileyo ukuxhuzula. Ukuba idosi yemihla ngemihla ichiza mkhulu kuno 1000 mg, kunye isilumkiso kufuneka uthathe zokucwangcisa ngomlomo. zingatshintshwa Le pharmacokinetics incindi yedlala phantsi kwempembelelo amayeza "Keppra".
Tablets "Keppra" bayakhuthazwa ukuba bathathe ungatyanga. nezinga kakhulu kuncitshiswa ukufakwa icandelo engundoqo esebenzayo xa kusetyenziswa emva za ulungisa ukutya.
Data ngokuphathelele intsebenziswano beziyobisi kunye notywala, akukho.
analogs
Ezikhemisti ezininzi kuThixo iziyobisi anticonvulsant ezikumgangatho ophezulu. Ngoko ke, ukuba amayeza ekunene lafunyanwa isela elo, ungasoloko ufumana i-analogu elungileyo. Yizani uncedo ugqirha kulo mbandela. Yena uya kukuxelela ukuba ngawaphi amayeza aya kusebenza kwityala elithile. Yamkelekile iziyobisi ethandwayo phakathi iingcali "Lamictal". Eyona nto iphambili esebenzayo i lamotrigine. Njengoko izinto abancedisayo benza monohydrate lactose, isodiyam carboxymethyl starch oxide intsimbi etyheli, nemagnesium stearate, kunye povidone. Ichiza abangaqeshwayo kwi nothomalaliso entsonkothileyo zezigulane sokuwa ezindala ngaphezu kweminyaka emi-3.
"Epiterra" iipilisi ezisetyenziswa kakhulu ekunyangeni ukuxhuzula. Kukwakho yengundoqo isithako levetiracetam esebenzayo. Njengoko excipients kusetyenziswa starch ingqolowa, isodiyam croscarmellose, povidone, nezinki stearate. Amayeza ezimiselweyo unyango izigulane abangaphezu kweminyaka elishumi. abantwana uthole kokuba contraindicated ngokungqongqo.
Izimvo amayeza "Keppra"
Izigulane sokuwa eyaziwa iziyobisi "Keppra". Izimvo namayeza unokuviwa emihle. Icandelo lokuqala esebenzayo kakhulu inegalelo ukunciphisa inani ukuxhuzula. Nangona kunjalo, ngexesha lokuqala unyango uyakwazi ukuphuhlisa iziphumo ebezingalindelekanga. Ba okwethutyana kwaye musa ukuba ukupheliswa unyango.
ukubuyekeza embi ngayo amayeza uninzi kwamatyala kwenzeka izigulane abo ngokwaneleyo yafunda imiyalelo. Idosi kufuneka ziqwalaselwe ngononophelo kwaye ingxelo nogqirha wakho malunga naluphi ukubonakalalisa basabele ezibi.
ukuthenga phi?
Le medicament inikwa ezikhemisti ezininzi. Oku wathengisa kuphela ngokumiselwa. Ngoko ke, akayi kuba kwenzeke ngaphandle kagqirha likagqirha ukuthenga elucwecweni okanye isisombululo. Xa zi-odola amayeza intanethi, iya kuba nako ukusindisa kakuhle. Kufuneka uhlawule malunga 900 engange nganye pack "Keppra" iipilisi. Imiyalelo yokusebenzisa, ukubuyekeza amayeza - konke oku kuxoxwe umphathi an kwikhemesti Internet.
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