ZempiloAmalungiselelo

Imiyalelo eneenkcukacha "Futsisa": ezibonisa ukusetyenziswa, analogs kunye nohlolo

Kunye arhente isibulala-zintsholongwane, arhente nokubola ngokuphumelelayo izigulane ukuphelisa izifo ezo zibangelwa amagciwane sengozini kubo into esebenzayo.

Okwangoku, kukho inani elikhulu kakhulu kumayeza anjalo. iimpawu zabo amayeza rhoqo idibana. Kodwa ke uninzi ziingcali amisele ichiza enjalo kwizigulane zabo "Futsis". Imiyalelo yokusebenzisa kunye neempawu zesixhobo kuya kwenziwa izinto kweli nqaku.

Ekwakhiweni, imilo kunye nokupakishwa

Ichiza "Futsis" imfundiso leyo elungiselwe yimfumba yekhadibhodi, zingathengwa ngohlobo iipilisi. isithako yabo esebenzayo usebenza njenge-fluconazole. Kwakhona kwi medicament nayo iquka amacandelo abancedisayo.

imveliso kujongwa eveliswe ngeedosi ka-50, 150, 100 no-200 mg. Amacwecwe isixa amaqhosha 4, zipakishwe khadibodi pack blister, ngokulandelelana.

Yiyiphi enye ifomu zingathengwa 'Futsis "? Imiyalelo yokusebenzisa (tablets - le ayilulo uhlobo kuphela lathi) ingxelo ukuba medicament yenziwa ngokohlobo isisombululo ukumnika. Ukubunjwa iquka amacwecwe fluconazole kunye izithako ezongezelelekileyo ezifana microcrystalline kwincindi, povidone K30, lactose, talc, nemagnesium stearate, isodiyam croscarmellose, sodium starch glycolate kunye nabanye.

Ewiliko for kwizitofu emthanjeni xa ithunyelwa iibhotile ml 100.

Ke ukuba ijeli "Futsis", ngoko ke ingathengwa zohlobo lwe-30 g

Pharmacology medicament

Ziziphi iinkalo ezendeleyo ichiza "Futsis 'na? imiyalelo Isicelo inikeza ukuba uthe kuthetha ifom ngamnye umsebenzi nokubola libizwe.

Fluconazole i yemvelaphi ezithambileyo bobabo kwiqela imichiza thiazole. Le nto inceda ukuphelisa umsebenzi enzymatic lwamacandelo ezithile leyo kwiiseli ezinzwaneni.

Emva ichiza aphazanyiswa kuyondelelaniswe yebhayoloji yolo iikhompawundi sterol kunye elinganeno kwinkqubo yokuguqulwa lanosterol ergosterol. utshintsho olunjalo inwebu yeseli ukukhuthaza ukumisa lokwanda nomngundo.

iimpawu ichiza

Yintoni iimpawu ichiza "Futsis"? Imiyalelo yokusebenzisa (iipilisi abe neempawu ezifanayo amayeza njengoko isisombululo kunye nejeli) uthi le zinetyhefu medicament iimpawu ephantsi. Kule nkalo, akukho nefuthe elibi emzimbeni womntu, kwakunye nefuthe elibonakalayo kubungakanani cytochromes kunye iihomoni androgenic kwi plasma yegazi.

Pharmacokinetics beziyobisi

Imiyalelo "Futsisa" uthi emva kokuthatha iipilisi ngaphakathi pretty ngokukhawuleza kwaye ako kakuhle iphecana zesisu. Ngokutsho iingcali, i-fluconazole sele bioavailability eliphezulu. Ukusetyenziswa ukutya alunasiphumo kwi inkqubo kukufakwa isixhobo.

Le xi ubuninzi into esebenzayo kwi plasma yegazi emsebenzini emva malunga 60-90 kwemizuzu emva nolawulo.

Kujongwa amayeza kakuhle waya ukwakhiwa neencindi zomzimba kunye namalaphu. Fluconazole sidlula kwi umqobo igazi-ingqondo kwaye bagxile kwi ulwelo lwe-cerebrospinal.

Kukhuthaza ichiza ivela emzimbeni wakhe oluqhutywa yokuchama. Bawo-ubomi imalunga 30 iiyure.

Ziziphi iparameters kwikinetiki na isisombululo "Futsis"? Guide ithi ukuba pharmacokinetics beziyobisi xa ilawulwa yegazi akukho eyahlukileyo kakhulu ukusuka kulawulo ngomlomo.

Ngokumalunga-arhente nokubola ngohlobo yejeli, oko neneempawu ezifanayo kunye nomsebenzi. gel ingakumbi ngempumelelo kuziveza xa dermatophytes kunye amagwele.

Nangona isicelo ngokwemixholo sixhobo, okuncinane arhente esebenzayo ongena egazini. Kule nkalo, akubikho ngokupheleleyo amanyathelo systemic.

Iingcali iye yafumanisa ukuba ijeli le ngokungalunganga ukuphembelela imeko yesikhumba.

Ubungqina obubonakalayo buxela

Imiyalelo "Futsisa" ingxelo ukuba ichiza isoloko isetyenziswa kunyango lwezifo ezosulelayo of eyendawo ezahlukahlukeneyo, nto leyo sabangela amagciwane, ebonisa uvakalelo oluphezulu ku-fluconazole. Njengomgaqo, iziyobisi ingqalelo amisiweyo gynecologists, dermatologists kunye mycologists.

Ngoko xa ukusebenzisa iziyobisi "Futsis" (tablets)? Guide ingxelo ukuba yemithi le fomu:

  • unyango mycosis, kwenzeka phezu iinyawo kunye nakummandla nasemiphakathweni, onychomycosis, ulwazi olusisikhokelo kunye olusisikhokelo versicolor;
  • usulelo lweenwebu yangaphakathi, apho zibangelwa fungi ze sodidi Candida;
  • izifo candidal yeendawo ezahlukeneyo (umz, candidemia, candidiasis zasasazwa, kunye nezinye iintlobo candidiasis candiduria ngokubanzi ukuba zibangelwa ngundo Candida);
  • izifo ayiphazamisi bronchopulmonary candidal;
  • unyango kweefom ezingapheliyo kunye nokoyika candidiasis lobufazi (yomhla nezolo);
  • candidiasis okondeleyo isifo somlomo, nto leyo enxulumene unxibe amazinyo;
  • unyango lwe histoplasmosis, sporotrichosis kunye nezinye mycoses ikho.

Yintoni injongo ukulungiselela ngomlomo "Futsis" (tablets) linokukwenziwa? Imiyalelo ithi ukuba ichiza isoloko isetyenziswa kuthintelo ukuphinda kwizigulane kunye:

  • balanitis candidal;
  • candidiasis ezingapheliyo zangasese;
  • izifo cryptococcal of eyendawo ezahlukeneyo;
  • izifo fungal of eyendawo ezahlukeneyo, ukuba isigulane unesifo immunodeficiency okanye ukufumana unyango cytostatic nemitha.

Ke ukuba isisombululo yolawulo iimela, lo myalelo "Futsisa" libonisa ukuba olu hlobo beziyobisi asetyenziswe kunyango:

  • cryptococcal meningitis;
  • izifo systemic ezinzwaneni (candidemia, usulelo lwamehlo candidal candiduria endocardium);
  • izifo cryptococcal esikhumba kunye isixokelelwano sokuphefumla.

Ichiza lokusebenza lwangaphandle ukuze yabelwe xa:

  • enesitshanguba ezibangela nagwele;
  • olusisikhokelo (jock nangenjinana, imbaleki kaThixo unyawo, trichophytosis, pityriasis versicolor kunye nosulelo kandidnyh).

Izimo

Yintoni irejimeni yonyango "Futsis" kweziyobisi abantwana? Guide ithi ukuba yindlela abadala kunye abantwana akukhuthazwa ukuba zisetyenziswe ubuntununtunu luyaphuculwa izinto ngamanye ichiza. Kwakhona alusetyenziselwa phambi aleji iikhompawundi azole ekufuphi kubume ku-fluconazole.

Sesikolweni xa engakanani ngobudala awazuze "Futsis DT 'abantwana? Imiyalelo usixelela ukuba la macwecwe eqhelekileyo ukuba contraindicated kakhulu ukuba unyango zabantwana ukuya kutsho kwiminyaka 7, wabathi saa - ukuya kwiminyaka emi-3.

amayeza Kwakhona kubhekwe Akuvunyelwe ukufumana ngethuba lokukhulelwa nokuncancisa. Oku ayisetyenziselwa unyango labantu abafumana unyango "cisapride" kunye "terfenadine" yaye abo umsebenzi zigazi enxulumene ulawulo ngeemoto ngoomatshini abayingozi.

Drug "Futsis DT": imiyalelo yokusebenzisa

Le medicament azipilisi, kwakunye isisombululo kunye gel kufuneka zisetyenziswe ngendlela eyahlukileyo.

Indlela ukuthatha ichiza "Futsis 50"? Manual ithi ukuba amayeza kunye isiqulatho into esebenzayo kwi 50-200 mg isetyenziselwa ukunyanga abantu abadala kuphela, kodwa izigulane abaselula iminyaka 3-7.

Iipilisi ziyathathwa naliphi na ixesha lemini ngomlomo. Idosi yemihla ngemihla ichiza ilungiselelwe ngexesha elinye kwaye ibekwe kuphela gqirha (kuxhomekeka phezu sifo).

Indlela yokusebenzisa le amacwecwe saa "Futsis" (50 mg)? Guide ingxelo ukuba ngaphambi kokuba eli chiza kufuneka unyityilikiswa emanzini eziqhelekileyo (5 ml).

Abantu abanengxaki candidiasis angasese, ichiza kanye ilawulwa emacwecweni 150 mg. Ukuthintela ukwenzeka candidiasis langasese uhlobo ezingapheliyo (thrush) iyeza lisetyenziswa idosi enye, kodwa kanye kuphela ngenyanga.

Ngokubanzi, indlela idosi azithathwa kuxhomekeke indlela isicelo wayo, kwaye akawatshintshi ngethuba lenguqu ukusuka kulawulo parenteral ukuya ngomlomo.

Umthamo isisombululo nokubandakanywa

Umyalelo "Futsisa" ithi kumalungiselelo isitofu efakwa iqulethe 200 mg i-fluconazole kunye 100 ml umxube sodium chloride (isotonic).

Phambi kokuba kuqaliswe medicament ukuba isigulane kufuneka ukusetyenziswa kuphela ngamanzi sodium. Kananjalo kufuneka ukuba siqwalasele isiqulatho chloride kesodiyam ion in isisombululo.

Nangona kungekho severe ukungavumelani lwemithi imali kufuneka ingabi ukuxutywa kunye nezinye iziyobisi ukumnika.

Ukusetyenziswa yejeli

Gel "Futsis" kwakunye iipilisi, kuyimfuneko ukusebenzisa kanye ngemini. I-arhente yangaphandle ngobunono atyabukile kwimimandla ulusu ochaphazelekayo, kwakunye kwimimandla ibekwe ngeenxa zonke.

Iingcali ingxelo yokuba ukuphumeza isiphumo isiqabu isigulana sidinga kuphela imali encinci gel. Lakhe wagcoba ngenyameko phesheya fungi yendawo kumphezulu ochaphazelekayo, ukwenzela ukuthintela maceration.

Ngoku uyazi ukuba mawuzisebenzise njani isisombululo gel kunye "Futsis" Amacwecwe (150 mg). Imiyalelo ithi ukuba idosi ixesha lokusebenzisa nganye iifomu ezithunyelwa kufuneka kumiselwa kuphela ngugqirha khona.

imiphumela emibi

Yintoni iziphumo ebezingalindelekanga kunokubangela ukusetyenziswa isisombululo iimela, gel kunye neepilisi "Futsis 150"? Umyalelo ithi ukuba imvelaphi ukusetyenziswa kwale mali, isigulane lisenokuba abasabela ezibi zilandelayo:

  • kakhulu yintloko, komhlaba, isiyezi kunye yombono;
  • arrhythmia kunye tachycardia;
  • isicaphucaphu, iintlungu esiswini, ukugabha, ukungacoleki kokutya, urhudo, kunye nezinye;
  • ziyabagulisa eluswini ngokohlobo alopecia, ityhefu epidermal necrosis, ukurhawuzelela, irhashalala, izigxala, nokudumba, Stevens-Johnson syndrome.

Kwakhona, ukusetyenziswa kwale iyeza kungachaphazela ukusebenza iimvavanyo laboratory (neutropenia, leukopenia, agranulocytosis, hypokalemia, thrombocytopenia, triglycerides kunye cholesterol egazini).

Ezi ziphumo bezingalindelekanga ifuna kumiwe ngoko nangoko "Futsisa".

amacala libanda

Kwimeko iipilisi "Futsis" libanda, okanye isisombululo isigulane lisenokuba ezinjalo iimpawu ezimbi ezifana nesiyezi, intloko ebuhlungu kunye nemibono. Ukongeza asikwazi, ngaphandle ukuziphatha usoyika.

Xa libanda kakhulu esiswini wahlamba kunye nonyango nomqondiso.

iyahambelana namanye amachiza

isicelo ngaxeshanye yesisombululo tablets 'Futsis "kunye anticoagulants inyusa ngokubonakalayo isiphumo yabo. Ngoko ke, ukubekwa esweni rhoqo lwezalathisi yexesha prothrombin.

amayeza ithatyathwa kungandisa lamanani plasma "benzodiazepines", "Midazolam", "Cyclosporin", "phenytoin" yaye "rifabutin 'egazini. Flucanozole Xa kudityaniswe nayiphi na kwezi ndlela kungafuna izilungiso zethamo mkhanya onamava specialist. Ukuba ngoyaba i data iingcebiso, efana ukuhlanganiswa kungandisa iziphumo ebezingalindelekanga reactions lengqondo unobangela nophuhliso njalo njalo.

Kunye nokusetyenziswa rhoqo hydrochlorothiazide with "Futsisom" ungalindela ukunyuka okubonakalayo igazi yoxinaniso ka-fluconazole. Noko ke, oku akuthethi kufuna uhlengahlengiso idosi.

Ukufumana iziyobisi bathi akusenzi yintshukumo zokucwangcisa ngomlomo ahlangeneyo.

Uthomalaliso "Futsisom" Izigulane abanesifo seswekile kufuneka athathe ingqalelo kuphuhliso Kusenokwenzeka hypoglycemia.

unyango ngaxeshanye nalo eli chiza, "rifampicin" ifuna ukwanda ithamo-fluconazole.

Indibaniso "Futsisa" yaye "Tacrolimus" ngokufuthi kakhulu kubangela ukwandiswa kwelifa nephrotoxicity yabo.

Ixabiso kunye analogue ze-arhente nokubola

Emva nokuqeshwa "Futsis" nokubola iziyobisi, izigulane ezininzi ukubuza malunga kubiza kangakanani. Kufuneka kuqatshelwe ukuba inani lamayeza ngamatyathanga kwikhemesti ezahlukeneyo zisenokuthi zahluke kancinane. avareji ixabiso layo malunga 300-400 engange (kungakhathaliseki uhlobo yokukhululwa).

Kuba iziyobisi, efanayo iimpawu amayeza ziquka iziyobisi ezifana "fluconazole", "Fukortsin", "Clotrimazole" yaye "Livarol". Noko ke, ngenxa yokwamkela yabo kufuneka bazi ukuba babe eyahlukileyo ngokupheleleyo iziphumo ebezingalindelekanga kunye Izimo. Ngoko ke, kufuneka usoloko udibane nogqirha ukubuyisela i "Futsisa" ngale ndlela. Hi ndlela leyi, imibutho yabasebenzi iza kukwazi ukukhetha i kwirejimeni echanekileyo nesebenza nezinyangayo.

Baqinisekiswa zee-arhente nokubola

Amaxesha amaninzi ingqalelo kulungiselelwa ukushiya ingxelo entle. Ngokutsho yakutshanje, Kuyinto ngokubanzi kusetyenziswa xa kusenziwa yamanina kwi unyango thrush. Noko ke, abantu abaninzi bathi arhente anti-ezinzwaneni "Futsis" kukwanceda ukuphelisa le sifo ebuhlungu kakhulu ixesha elide. Noko ke, iingcali ingxelo ukuba umntu silibale ngayo amanye amayeza zinceda ukubuyisela izilwanyana abaqhelekileyo kwi lobufazi.

Ethetha ukusebenza "Futsis" iziyobisi, singasathethi ingxelo embi. Ezinye izigulane ziphathwa eli chiza, bathi ukutya iipilisi okanye ukusetyenziswa isisombululo baphawula iziphumo ebezingalindelekanga. Ngenxa umthetho, ukuba kuvela ukudumba, ukurhawuzelela, kwiinwebu impumlo kunye namehlo, nangecesina, intloko ebuhlungu kakhulu.

Ke ukuba ijeli "Futsis", i-ncomo ngayo azixhaphakanga. Xa kwabo, ngokutsho ukusebenza ephezulu kwesi sixhobo, ingakumbi unyango olusisikhokelo.

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