ZempiloAmalungiselelo

Codeine phosphate: imiyalelo ukusetyenziswa, analogs kunye nohlolo

Codeine bobabo umlaliso sezakhi series. Isetyenziswa ngokubanzi amayeza njengeyeza for khohlo. Libhekisela iyeza kundlunkulu acting leyo isoloko isetyenziswa ngokudityaniswa nezinye izinto, phakathi ezo ukuphilisa terpin. Kakhulu umdla kukuba ukusetyenziswa codeine ngazo iimpawu ukunxila okanye iziyobisi. imiphumela eziqwalaselweyo iintlungu. Kulo mba, codeine phosphate ingasetyenziswa njengento ndindisholo, kodwa ngokungqongqo ngokumiselwa.

ulwazi oluncincane

Umgaqo tyando ifana kakhulu codeine ku icaffeine. Nakuba kunjalo, iziphumo zayo iintlungu thile buthathaka. Kunye nale phosphate codeine (Latin kubonisa ekhobokisayo njengoko codeinum) anazo zomlomo ngamandla ukukwazi ukuthoba iziko ukhohlokhohlo excitation. Ukuqhubeka umzekeliso morphine, umzekelo, ukuba ngaphantsi ngxelo imbi kangaka kakhulu ukuphefumla kwabantu, kwaye hayi abangaphangeliyo umsebenzi iphecana zesisu. Ngaphandle koku, ngokufuthi kukho iimeko apho ichiza kunempembelelo oluvuselela emzimbeni, ukuvimbela ukozela.

Codeine phosphate: Inkcazo Izimo

Kanye eminye imithi, codeine ine uluhlu khorwisaka Izimo. Kufuneka bazi ngokuqinisekileyo ngaphambi kokuba usebenzise iziyobisi. Ukuze kuphuculwe imbono yakho, siye angamvaleli kuluhlu eyahlukileyo. Ngenxa yoko, ichiza kufuneka isetyenziswe phambi kwezi zinto zilandelayo:

  • hypersensitivity High;
  • arrhythmia;
  • ukuzibulala;
  • iingxaki isisu, prostate kunye urethra;
  • ekhulelwe okanye zisanyisa;
  • abadala okanye yobudala yabantwana;
  • Kuxhomekeka ekufumanekeni iziyobisi ichiza ekuthiwa phosphate codeine;
  • sorhudo;
  • iingxaki yokunxila;
  • dispensiya ubuthi;
  • ubukho ukuhlaselwa sisifo sombefu inyumoniya;
  • umonzakalo ebuchotsheni, kwakunye kwezintso okanye isibindi ukusilela.

Njengoko ubona, uluhlu mkhulu kakhulu. Ngokubanzi, phambi kokuba ukusetyenziswa codeine kufuneka ukuba udibane nogqirha wakho. Uyakukumisela imithi kuyimfuneko ukuba imeko emzimbeni wakho ikuvumela ukuba ukuthatha eli yeza.

Codeine phosphate: ukuthatha yaye yintoni ngokwemithamo njani?

Xa usebenzisa codeine ukulungiselela iinjongo zonyango kufuneka balumke ngokukodwa xa kuyilwa idosi echanekileyo kweziyobisi, kwakunye nexesha wokwamkelwa kwakhe. Ngoko ke, ukuba ahlekise kucetyiswa ukuba abadala ukuba 15-60 mg qho kwiiyure 3-6. Xa utyatyazo kuyehla kube umthamo 30 mg kane ngemini. Ekugqibeleni, xa uhlaselwe ukhohlokhohlo kufuneka asele 10-20 mg beziyobisi amaxesha-4 ngemini. umthamo Higher yemihla ngemihla ye-codeine phosphate elithe (kufuneka ubhale nogqirha amayeza) yi-120 mg.

Ngokuba abantwana umthamo kancinci eyahlukileyo. Ngokuqhelekileyo, lo mlinganiselo phandle 0.5 mg nganye 1 kg ubunzima bomzimba, xa kufikwa abathintela iintlungu ezahlukeneyo. Xa ukhohlela kufuneka ukuba uthathe mg ngaphezulu kwama-15. Ekugqibeleni, ne sorhudo njengoko idosi ichanekile 0.5 mg ngamnye 1 kg ubunzima bomzimba. Malunga nezihlandlo reception, oko kukuthi, njengokuba abadala, kufuneka ilingane amaxesha 4-5 ngosuku. Hi ndlela leyi, abantwana abangaphantsi abafumana codeine phosphate ayikhuthazwa kwiminyaka emi-2.

imiphumela kwemithi

Njengoko kukhankanyiwe ngaphambili, codeine i antitussive embindini olibambela. Ku fanele ku sezakhi phenanthrene lwe thotho. Ngaphezu koko, oko kunxulumene agonists opioid receptor enokuthi kakhulu ekunciphiseni excitability lweziko ukukhohlela, ngenxa inhibition yayo ngqo. umsebenzi iintlungu unokucacisa kweziyobisi ukusebenza receptors opiate ebonisa excitation kwiindawo ezininzi nkqubo luvo. Plus, oko litshintsha inani umbono ngokweemvakalelo intlungu. Ngokubanzi, ibonisa ukuba isiphumo iintlungu ngokwayo emva kwemizuzu 10-45 emva kokuba isitofu, yaye nge kangangesiqingatha seyure xa usebenzisa iipilisi codeine phosphate. Ubude amanyathelo yoviwo ithatha malunga neeyure ezi-4.

imiphumela emibi

Kakade ke, codeine phosphate lineziphumo zalo ezisemacaleni, apho wonke umntu ngazo ngeendlela ezahlukeneyo. Njengoko kwimeko Izimo, siya kumnika uluhlu neziphumo bavame emva kokusebenzisa le nto:

  • I-luvo nga lokuwela senzo: ukwanda ukozela, ebuhlungu kunye nesiyezi (kunqabile), kungenzeka ukuba nemibono okanye babebona ezibonwayo, ixhala, amabi zibe amaphupha, ukudandatheka (kwisehlo enqabileyo), kwakunye ukuxhuzula. Xa ukusetyenziswa amathamo ngokugqithisileyo bangafumana iingcangcazela, ukonakala uququzelelo ngeemoto ngqongqo kwezihlunu.
  • Kwinkqubo yokwetyisa, ezi ziphumo zilandelayo: isicaphucaphu nokugabha (ngamaxesha ambalwa), ukuqhina, amahlaba esiswini, umlomo owomileyo, kungenzeka ukuba uneanorexia kwaye, ekugqibeleni, hepatotoxicity.
  • inkqubo Cardio nemithambo: arrhythmia, ukuncipha ngesiquphe okanye ukunyuka koxinzelelo lwegazi.
  • isixokelelwano sokuphefumla: inhibition elinqatyisiweyo leziko zemiphunga okanye atelectasis.
  • Kukho kwakhona okuba le negazi zilandelayo: amaqhakuva, iindumbisa ubuso nasemqaleni, ukurhawuzelela, bronchospasm, laryngospasm, kunye urticaria.
  • Ukuba ezinye iziphumo ebezingalindelekanga ezivela ekusetyenzisweni codeine phosphate (isiLatin, ngokuzenzekelayo, izandi codeinum) ziquka ukubila ngokugqithiseleyo, chaza luncinane euphoric. Kwakunye ingozi ukuxhomekeka kunye ezinde yokusebenzisa (ingakumbi ezininzi).

Kakade ke, ingozi iziphumo ebezingalindelekanga ngentla okhankanywe lincinane kakhulu. Ewe, yaye ngokufuthi ziyahluka ukusuka inyathelo kwisenzo.

iimpawu libanda

ziquka Iimpawu ngezenzeko ilandelayo libanda ezigulo ezondeleyo: ukudideka kwengqondo, isiyezi kakhulu, uvalo kunye ndlongo, unditsho, ubuthathaka jikelele yokusithwa lomzimba kunye noxinzelelo lwegazi. Kwiimeko kakhulu, kukho amathuba aphezulu yokulahlekelwa sezingqondweni okanye ukuba khokhoma ukuqala. unyango mkhuba okanye libanda, kunokuba kakhulu elide yaye kungabi lula. Kwiimeko ubuthi kufuneka iphume nesisu, ukubamba umoya wakhe ukuxhasa umsebenzi intliziyo. Kwezinye iimeko, kusengqiqweni ukuba isitofu naloxone, nto leyo ochasene ethile analgesics opioid.

imiyalelo Special ngexesha unyango

Xa kukho inkqubo lokubuyisela emva codeine libanda, okanye unyango ngale ngxaki yakhe, izigulane kufuneka uyeke ukusela utywala. Inyaniso kukuba ngexesha unyango ebantwini buthuntu noko kujoliswe kunye nesantya ngayo lengqondo. Utywala ukuze sibe sibi eyomeleleyo kuphela. Kwaye kungaba nefuthe elibi umntu ekwenzeni imisebenzi enokubakho eyingozi.

Oku kufuna ingqalelo ekhethekileyo ngethuba lokukhulelwa kwabasetyhini. Eneneni, ukusetyenziswa codeine kungabangela ukulibaziseka Ukuqina, yaye ngamanye amaxesha unikezelo ngokukhawuleza - isongezo. Ngokubanzi, iziqhulo kokubi. Ekugqibeleni, njengoko kutshiwo apha ngasentla, abantwana abaselula, ngokubanzi, kufuneka ukuba uthathe codeine. Kulo mzekelo, kukho amathuba enkulu ingenzeka of reactions ngamazwi, njengoko abantwana baye banda uvakalelo kwimiphumo analgesics opioid.

semthethweni

ERashiya, ngoku kukho ityala, usebenza Narcotics codeine. Ngoko ke, uyithenge ekhemesti ngaphandle kokumiselwa ayikwazi ukuba. Kutshanje, ukusetyenziswa inkcubeko codeine waqalisa ukulumkisa uluntu, njengoko ukwanda ichiza ikhula ngokucacileyo. Ngeendlela ezininzi oku "emagqabini" yala magcisa hip-hop yaseMelika abadla uNojaji ukusetyenziswa Purple abanxilileyo - ukusela okhethekileyo equlathe amathamo eliphezulu codeine. isiraphu kwegunya bomvu-nemfusa eziyiyo yaye kutheni igama engaqhelekanga enjalo. Emva ukusela ulwelo, uya udibana imvakalelo imincili ezingephi ezifanayo bethabatheke kunye opiates, leyo, enyanisweni, ibhekisela codeine. Songs of rap American badla ungaqulatha umbhalo, isalatha kulaa ukusetyenziswa eyondeleleneyo Purple abanxilileyo. Hi ndlela leyi, umdali le intshukumo - Dj Screw. Yena wafa eneminyaka engama-29 ukusuka libanda kakhulu codeine.

Kufuneka kuqatshelwe ukuba codeine afumaneka kwezinye amayeza, kubandakanywa zonke iintlobo ifiva, protivomigrenoznye kunye nabanye. Kulo mba, iziyobisi abaninzi baye wavalwa ezithengiswayo kummandla Russia. Yaye ukwabiwa mthethweni kunye nokuthengiswa kunokuba ukufumana ukuya kwiminyaka eli-12 entolongweni.

Ekuphetheni

Codeine abe umda obanzi, njengoko imiphumela yayo emzimbeni womntu womelele kakhulu. Kusenokuba ngexeshana olude elifutshane ixesha ukutshintsha imbono somzimba yomntu. Eyona ndlela iqhelekileyo codeine (phosphate) - ngumgubo apho lula enyibilikayo emanzini. Ngenxa kwiipropati lalo, liye lasetyenziswa ngokubanzi amayeza. Noko ke, njengoko kusoloko kunjalo opiates, iyeza langena ngokukhawuleza ezitratweni, nto leyo iba nefuthe elibi kubantu odlayo kuwo, imiphumo ngisho lingakubulala.

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